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TargetVasopressin V1b receptor(Rat)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50205313(d[Leu4]AVP | CHEMBL265859)
Affinity DataKi:  0.0400nMAssay Description:Displacement of [3H]AVP from rat vasopressin V1b receptor expressed in At-T20 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Rat)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50205305(d[Arg4]AVP | CHEMBL375324)
Affinity DataKi:  0.130nMAssay Description:Displacement of [3H]AVP from rat vasopressin V1b receptor expressed in At-T20 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Rat)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50205309(d[Leu4,Lys8]VP | CHEMBL412972)
Affinity DataKi:  0.160nMAssay Description:Displacement of [3H]AVP from rat vasopressin V1b receptor expressed in At-T20 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Rat)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50205296(d[Arg4,Dab8]VP | CHEMBL385739)
Affinity DataKi:  0.190nMAssay Description:Displacement of [3H]AVP from rat vasopressin V1b receptor expressed in At-T20 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Rat)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50205291((S)-1-((4R,7S,10S,13S,16S)-7-(2-amino-2-oxoethyl)-...)
Affinity DataKi:  0.200nMAssay Description:Displacement of [3H]AVP from rat vasopressin V1b receptor expressed in At-T20 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Rat)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM35667([3H]Argipressin tannate | AVP | [3H]Arginine vasop...)
Affinity DataKi:  0.230nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2012
Entry Details
PubMed
TargetVasopressin V1b receptor(Rat)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50205297(d[Leu4,Dab8]VP | CHEMBL412973)
Affinity DataKi:  0.25nMAssay Description:Displacement of [3H]AVP from rat vasopressin V1b receptor expressed in At-T20 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Rat)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50205300(d[Val4]AVP | CHEMBL221436)
Affinity DataKi:  0.25nMAssay Description:Displacement of [3H]AVP from rat vasopressin V1b receptor expressed in At-T20 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Rat)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50205301(d[Leu4,Orn8]VP | CHEMBL375188)
Affinity DataKi:  0.260nMAssay Description:Displacement of [3H]AVP from rat vasopressin V1b receptor expressed in At-T20 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Rat)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50205303(d[Leu4,Dap8]VP | CHEMBL373968)
Affinity DataKi:  0.380nMAssay Description:Displacement of [3H]AVP from rat vasopressin V1b receptor expressed in At-T20 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Rat)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50205306(d[Orn4,Lys8]VP | CHEMBL375323)
Affinity DataKi:  0.450nMAssay Description:Displacement of [3H]AVP from rat vasopressin V1b receptor expressed in At-T20 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Rat)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50205311(d[Orn4]AVP | CHEMBL375096)
Affinity DataKi:  0.450nMAssay Description:Displacement of [3H]AVP from rat vasopressin V1b receptor expressed in At-T20 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Rat)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50205292(d[Arg4,Orn8]VP | CHEMBL385068)
Affinity DataKi:  0.600nMAssay Description:Displacement of [3H]AVP from rat vasopressin V1b receptor expressed in At-T20 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Rat)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50205298(d[Arg4,Lys8]VP | CHEMBL375325)
Affinity DataKi:  0.600nMAssay Description:Displacement of [3H]AVP from rat vasopressin V1b receptor expressed in At-T20 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
TargetVasopressin V1a/V1b receptor(Rat)
Albert Szent-Gy£Rgyi Medical University

Curated by ChEMBL
LigandPNGBDBM35667([3H]Argipressin tannate | AVP | [3H]Arginine vasop...)
Affinity DataKd:  0.650nMAssay Description:Compound was evaluated for its dissociation constant (Kd) to rat liver Vasopressin V1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/30/2012
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Rat)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50205307(d[Cha4,Dab8]VP | CHEMBL412742)
Affinity DataKi:  0.800nMAssay Description:Displacement of [3H]AVP from rat vasopressin V1b receptor expressed in At-T20 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Rat)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50205310(d[Orn4,Orn8]VP | CHEMBL219272)
Affinity DataKi:  0.910nMAssay Description:Displacement of [3H]AVP from rat vasopressin V1b receptor expressed in At-T20 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Rat)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50299343(SSR149415 | (2S,4R)-1-[5-Chloro-1-[(2,4-dimethoxyp...)
Affinity DataKi:  1nMAssay Description:Displacement of [3H]Arg8-vasopressin from rat vasopressin V1b receptor expressed in CHO-K1 cells by Packard Topcount scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2012
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Rat)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50299343(SSR149415 | (2S,4R)-1-[5-Chloro-1-[(2,4-dimethoxyp...)
Affinity DataKi:  1nMAssay Description:Displacement of [3H]AVP from rat vasopressin V1b receptor expressed in CHO cells by whole cell binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Rat)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50299343(SSR149415 | (2S,4R)-1-[5-Chloro-1-[(2,4-dimethoxyp...)
Affinity DataKi:  1.30nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/3/2012
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Rat)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50205312(d[Cha4]AVP | CHEMBL265858)
Affinity DataKi:  1.40nMAssay Description:Displacement of [3H]AVP from rat vasopressin V1b receptor expressed in At-T20 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Rat)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50205293(d[Cha4,Lys8]VP | CHEMBL221485)
Affinity DataKi:  1.90nMAssay Description:Displacement of [3H]AVP from rat vasopressin V1b receptor expressed in At-T20 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
TargetVasopressin V1a/V1b receptor(Rat)
Albert Szent-Gy£Rgyi Medical University

Curated by ChEMBL
LigandPNGBDBM50137948(Biphenyl-2-carboxylic acid [2-[3-(4-methyl-[1,4]di...)
Affinity DataIC50: 2nMAssay Description:Inhibitory activity against arginine vasopressin V1 receptor using [3H]AVP as radioligand in rat liverMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Rat)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50338810(N-isopropyl-2-(2-(3-methoxyphenyl)-4-oxo-6-(3-(pip...)
Affinity DataIC50: 2nMAssay Description:Displacement of [3H]AVP from rat vasopressin V1b receptor expressed in CHO cells by whole cell binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Rat)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50205295(d[Cha4,Orn8]VP | CHEMBL263090)
Affinity DataKi:  3nMAssay Description:Displacement of [3H]AVP from rat vasopressin V1b receptor expressed in At-T20 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
TargetVasopressin V1a/V1b receptor(Rat)
Albert Szent-Gy£Rgyi Medical University

Curated by ChEMBL
LigandPNGBDBM50137945(Biphenyl-2-carboxylic acid [2-[4-(4-methyl-piperaz...)
Affinity DataIC50: 3nMAssay Description:Inhibitory activity against arginine vasopressin V1 receptor using [3H]AVP as radioligand in rat liverMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Rat)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50299343(SSR149415 | (2S,4R)-1-[5-Chloro-1-[(2,4-dimethoxyp...)
Affinity DataKi:  3.70nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/3/2012
Entry Details Article
PubMed
TargetVasopressin V1a/V1b receptor(Rat)
Albert Szent-Gy£Rgyi Medical University

Curated by ChEMBL
LigandPNGBDBM50075816(Mca1,D-Trp2,Sar7AVT | CHEMBL264208)
Affinity DataKd:  3.80nMAssay Description:Compound was evaluated for its dissociation constant (Kd) to rat liver Vasopressin V1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/30/2012
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Rat)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50338811(2-(2-(3-chlorophenyl)-4-oxo-6-(3-(piperidin-1-yl)p...)
Affinity DataIC50: 4nMAssay Description:Displacement of [3H]AVP from rat vasopressin V1b receptor expressed in CHO cells by whole cell binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetVasopressin V1a/V1b receptor(Rat)
Albert Szent-Gy£Rgyi Medical University

Curated by ChEMBL
LigandPNGBDBM50137953(Biphenyl-2-carboxylic acid [2-[4-(4-diethylamino-p...)
Affinity DataIC50: 4nMAssay Description:Inhibitory activity against arginine vasopressin V1 receptor using [3H]AVP as radioligand in rat liverMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V1a/V1b receptor(Rat)
Albert Szent-Gy£Rgyi Medical University

Curated by ChEMBL
LigandPNGBDBM50137940(Biphenyl-2-carboxylic acid [2-[4-(4-dimethylamino-...)
Affinity DataIC50: 6nMAssay Description:Inhibitory activity against arginine vasopressin V1 receptor using [3H]AVP as radioligand in rat liverMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V1a/V1b receptor(Rat)
Albert Szent-Gy£Rgyi Medical University

Curated by ChEMBL
LigandPNGBDBM50291329(8-arginine vasopressin trisulphide | CHEMBL267405)
Affinity DataIC50: 9.5nMAssay Description:Tested for the TYR(Me)2 arginine-vasopressin as radioligand at 0.3 nM in A7r5 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetVasopressin V1b receptor(Rat)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50205299(d[Cha4,Dap8]VP | CHEMBL375187)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]AVP from rat vasopressin V1b receptor expressed in At-T20 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
TargetVasopressin V1a/V1b receptor(Rat)
Albert Szent-Gy£Rgyi Medical University

Curated by ChEMBL
LigandPNGBDBM35667([3H]Argipressin tannate | AVP | [3H]Arginine vasop...)
Affinity DataIC50: 10nMAssay Description:Tested for the TYR(Me)2 arginine-vasopressin as radioligand at 0.3 nM in A7r5 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetVasopressin V1b receptor(Rat)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50299342(CHEMBL1204403 | CHEMBL1204126 | CHEMBL572709 | N-(...)
Affinity DataKi:  16nMAssay Description:Displacement of [3H]Arg8-vasopressin from rat vasopressin V1b receptor expressed in CHO-K1 cells by Packard Topcount scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2012
Entry Details Article
PubMed
TargetVasopressin V1a/V1b receptor(Rat)
Albert Szent-Gy£Rgyi Medical University

Curated by ChEMBL
LigandPNGBDBM50075817(Mpa-Car-lle-Gln-Asn-Cys-Sar-Arg-Gly-NH2 | CHEMBL23...)
Affinity DataKd:  17.8nMAssay Description:Compound was evaluated for its dissociation constant (Kd) to rat liver Vasopressin V1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/30/2012
Entry Details Article
PubMed
TargetVasopressin V1a/V1b receptor(Rat)
Albert Szent-Gy£Rgyi Medical University

Curated by ChEMBL
LigandPNGBDBM50075817(Mpa-Car-lle-Gln-Asn-Cys-Sar-Arg-Gly-NH2 | CHEMBL23...)
Affinity DataKd:  18nMAssay Description:Compound was evaluated for its dissociation constant (Kd) to rat liver Vasopressin V1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/30/2012
Entry Details Article
PubMed
TargetVasopressin V1a/V1b receptor(Rat)
Albert Szent-Gy£Rgyi Medical University

Curated by ChEMBL
LigandPNGBDBM50137942(Biphenyl-2-carboxylic acid [2-(4-[1,4']bipiperidin...)
Affinity DataIC50: 20nMAssay Description:Inhibitory activity against arginine vasopressin V1 receptor using [3H]AVP as radioligand in rat liverMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V1a/V1b receptor(Rat)
Albert Szent-Gy£Rgyi Medical University

Curated by ChEMBL
LigandPNGBDBM50137949(Biphenyl-2-carboxylic acid [2-[4-(4-methyl-[1,4]di...)
Affinity DataIC50: 20nMAssay Description:Inhibitory activity against arginine vasopressin V1 receptor using [3H]AVP as radioligand in rat liverMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V1a/V1b receptor(Rat)
Albert Szent-Gy£Rgyi Medical University

Curated by ChEMBL
LigandPNGBDBM50137956(Biphenyl-2-carboxylic acid [2-[4-(4-methyl-piperaz...)
Affinity DataIC50: 20nMAssay Description:Inhibitory activity against arginine vasopressin V1 receptor using [3H]AVP as radioligand in rat liverMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V1a/V1b receptor(Rat)
Albert Szent-Gy£Rgyi Medical University

Curated by ChEMBL
LigandPNGBDBM50137946(Biphenyl-2-carboxylic acid [2-[2-(4-dimethylamino-...)
Affinity DataIC50: 20nMAssay Description:Inhibitory activity against arginine vasopressin V1 receptor using [3H]AVP as radioligand in rat liverMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V1a/V1b receptor(Rat)
Albert Szent-Gy£Rgyi Medical University

Curated by ChEMBL
LigandPNGBDBM50137951(Biphenyl-2-carboxylic acid [2-{4-[(2-dimethylamino...)
Affinity DataIC50: 20nMAssay Description:Inhibitory activity against arginine vasopressin V1 receptor using [3H]AVP as radioligand in rat liverMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Rat)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50299342(CHEMBL1204403 | CHEMBL1204126 | CHEMBL572709 | N-(...)
Affinity DataKi:  21nMAssay Description:Displacement of [3H]Arg8-vasopressin from rat vasopressin V1b receptor expressed in CHO-K1 cells by Packard Topcount scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2012
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Rat)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50299349(1-(2-(1-(2,4-dimethoxyphenylsulfonyl)-1,2,3,4-tetr...)
Affinity DataKi:  23nMAssay Description:Displacement of [3H]Arg8-vasopressin from rat vasopressin V1b receptor expressed in CHO-K1 cells by Packard Topcount scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2012
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Rat)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM85094(NSC_64759 | CAS_62357-86-2 | dDAVP)
Affinity DataKi:  25.1nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2012
Entry Details
PubMed
TargetVasopressin V1a/V1b receptor(Rat)
Albert Szent-Gy£Rgyi Medical University

Curated by ChEMBL
LigandPNGBDBM50016310(CHEMBL406303 | [Mpa1Val4Sar7]AVP (Arginine-vasopre...)
Affinity DataKd:  27nMAssay Description:Binding affinity against plasma membrane from rat liverMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Rat)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50299358(1-(2-(1-(2,4-dimethoxyphenylsulfonyl)-1,2,3,4-tetr...)
Affinity DataKi:  27nMAssay Description:Displacement of [3H]Arg8-vasopressin from rat vasopressin V1b receptor expressed in CHO-K1 cells by Packard Topcount scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2012
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Rat)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM85096(NSC_105077 | CAS_105077 | d(CH2)5Tyr(Me)AVP)
Affinity DataKi:  37.6nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2012
Entry Details
PubMed
TargetVasopressin V1b receptor(Rat)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50013775(1-[19-Amino-13-sec-butyl-10-(2-carbamoyl-ethyl)-7-...)
Affinity DataKi:  39.4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2012
Entry Details
PubMed
TargetVasopressin V1a/V1b receptor(Rat)
Albert Szent-Gy£Rgyi Medical University

Curated by ChEMBL
LigandPNGBDBM50016310(CHEMBL406303 | [Mpa1Val4Sar7]AVP (Arginine-vasopre...)
Affinity DataKd:  42nMAssay Description:Binding affinity against plasma membrane from rat liver using [3H]-AVP as a radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
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