Compile Data Set for Download or QSAR
Report error Found 127 of affinity data for UniProtKB/TrEMBL: P54833
TargetBeta-2 adrenergic receptor(Dog)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM25392(Isoproterenol,(+) | CHEMBL434 | 4-[1-hydroxy-2-(pr...)
Affinity DataIC50: 0.100nMAssay Description:Agonistic activity for Beta-2 adrenergic receptor was assessed by it's inhibitory effect on spontaneous contractions in isolated rat uterusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2012
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Dog)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM25392(Isoproterenol,(+) | CHEMBL434 | 4-[1-hydroxy-2-(pr...)
Affinity DataIC50: 0.100nMAssay Description:Agonistic activity towards beta-2 adrenoceptor. IC50, the mean concentration required to produce 50% inhibition of uterine contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Dog)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM25761(Propanolol,(+/-) | PROPRANOLOL, l- | PROPRANOLOL,(...)
Affinity DataKd:  1.78nMAssay Description:Compound was evaluated for competitive antagonism of beta-2 adrenergic receptor in rat uterus measured as pA2 (-log KB)More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetBeta-2 adrenergic receptor(Dog)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50405147(4-Hydroxy Propranolol | 4-HYDROXYPROPRANOLOL SULFA...)
Affinity DataKd:  2.40nMAssay Description:Compound was evaluated for competitive antagonism of beta-2 adrenergic receptor in rat uterus measured as pA2 (-log KB)More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Dog)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50086666(8-(3-tert-Butylamino-2-hydroxy-propoxy)-4-{3-[4-(2...)
Affinity DataKi:  2.70nMAssay Description:Beta-2 adrenergic receptor binding affinity by measuring the displacement of [3H]DHA binding in rat lungMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Dog)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50002133((4-{2-[2-(3-Chloro-phenyl)-2-hydroxy-ethylamino]-p...)
Affinity DataIC50: 9.10nMAssay Description:Agonistic activity for Beta-2 adrenergic receptor was assessed by it's inhibitory effect on spontaneous contractions in isolated rat uterusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2012
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Dog)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM25761(Propanolol,(+/-) | PROPRANOLOL, l- | PROPRANOLOL,(...)
Affinity DataIC50: 17nMAssay Description:Tested for Beta-2 adrenergic receptor selectivity in canine lung tissue in anesthetized dogsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetBeta-2 adrenergic receptor(Dog)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50086673(8-(3-tert-Butylamino-2-hydroxy-propoxy)-4H-benzo[1...)
Affinity DataKi:  23nMAssay Description:Beta-2 adrenergic receptor binding affinity by measuring the displacement of [3H]DHA binding in rat lungMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Dog)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50405146(CHEMBL171432)
Affinity DataKd:  29.5nMAssay Description:Compound was evaluated for competitive antagonism of beta-2 adrenergic receptor in rat uterus measured as pA2 (-log KB)More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Dog)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50087518(6-fluoronorepinehprine | (R)4-(2-Amino-1-hydroxy-e...)
Affinity DataKi:  67nMAssay Description:Binding of [3H]dihydroalprenolol to beta-2 adrenergic receptor of rat cerebral cortical membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Dog)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50086670(8-{2-Hydroxy-3-[4-(2-methoxy-phenyl)-piperazin-1-y...)
Affinity DataKi:  88nMAssay Description:Beta-2 adrenergic receptor binding affinity by measuring the displacement of [3H]DHA binding in rat lungMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Dog)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50087520((R)3-Fluoro-4-(1-hydroxy-2-methylamino-ethyl)-benz...)
Affinity DataKi:  110nMAssay Description:Binding of [3H]dihydroalprenolol to beta-2 adrenergic receptor of rat cerebral cortical membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Dog)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50019060(CHEMBL287587 | 4-(2-Amino-1-hydroxy-ethyl)-3-fluor...)
Affinity DataKi:  140nMAssay Description:Binding of [3H]dihydroalprenolol to beta-2 adrenergic receptor of rat cerebral cortical membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Dog)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50019059(3-Fluoro-4-(1-hydroxy-2-methylamino-ethyl)-benzene...)
Affinity DataKi:  260nMAssay Description:Binding of [3H]dihydroalprenolol to beta-2 adrenergic receptor of rat cerebral cortical membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Dog)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50010834(CHEMBL98975 | 1-{2-[4-(3H-Imidazol-1-yl)-phenoxy]-...)
Affinity DataIC50: 280nMAssay Description:Tested for Beta-2 adrenergic receptor selectivity in canine lung tissue in anesthetized dogsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2012
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Dog)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50010840(CHEMBL421005 | 1-{2-[4-(3H-Imidazol-1-yl)-phenoxy]...)
Affinity DataIC50: 510nMAssay Description:Tested for Beta-2 adrenergic receptor selectivity in canine lung tissue in anesthetized dogsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2012
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Dog)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50122649((2-Chloro-4-{2-[2-hydroxy-2-(4-hydroxy-phenyl)-1-m...)
Affinity DataIC50: 525nMAssay Description:Agonistic activity for Beta-2 adrenergic receptor was assessed by it's inhibitory effect on spontaneous contractions in isolated rat uterusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2012
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Dog)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50001906(CHEMBL349978 | 4-Methanesulfonylamino-N-[4-(2-meth...)
Affinity DataIC50: 630nMAssay Description:Binding affinity towards Beta-2 adrenergic receptor by displacing [3H]dihydroalprenolol, in partially purified membrane fractions from canine lung ti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Dog)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50029050(4-[(1R)-1-hydroxy-2-(methylamino)ethyl]benzene-1,2...)
Affinity DataKi:  660nMAssay Description:Binding of [3H]dihydroalprenolol to beta-2 adrenergic receptor of rat cerebral cortical membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetBeta-2 adrenergic receptor(Dog)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50086664(8-{3-[4-(Furan-2-carbonyl)-piperazin-1-yl]-2-hydro...)
Affinity DataKi: >1.00E+3nMAssay Description:Beta-2 adrenergic receptor binding affinity by measuring the displacement of [3H]DHA binding in rat lung; Not Active means Ki >1000 nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Dog)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50086675(8-{3-[4-(4-Fluoro-benzoyl)-piperazin-1-yl]-2-hydro...)
Affinity DataKi: >1.00E+3nMAssay Description:Beta-2 adrenergic receptor binding affinity by measuring the displacement of [3H]DHA binding in rat lung; Not Active means Ki >1000 nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Dog)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50086660(6-{3-[4-(4-Fluoro-benzoyl)-piperazin-1-yl]-2-hydro...)
Affinity DataKi: >1.00E+3nMAssay Description:Beta-2 adrenergic receptor binding affinity by measuring the displacement of [3H]DHA binding in rat lung; Not Active means Ki >1000 nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Dog)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50773(1-[4-(2-methoxyphenyl)piperazin-1-yl]-3-naphthalen...)
Affinity DataKi:  1.00E+3nMAssay Description:Beta-2 adrenergic receptor binding affinity by measuring the displacement of [3H]DHA binding in rat lungMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Dog)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50014154(CHEMBL38465 | 2-(5-Methyl-1H-imidazol-4-ylmethyl)-...)
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity for Beta adrenergic receptor was determined by using [3H]dihydroalprenolol as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2012
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Dog)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50001900(CHEMBL162182 | N-{4-[(4-Phenyl-piperazin-2-ylmethy...)
Affinity DataIC50: 1.00E+3nMAssay Description:Binding affinity towards Beta-2 adrenergic receptor by displacing [3H]dihydroalprenolol, in partially purified membrane fractions from canine lung ti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Dog)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM25392(Isoproterenol,(+) | CHEMBL434 | 4-[1-hydroxy-2-(pr...)
Affinity DataIC50: 1.00E+3nMAssay Description:Compound was evaluated for its binding affinity towards beta-2 adrenergic receptor in rat soleus membrane by displacing (-)-isoproterenol (50 uM)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Dog)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50086674(6-{3-[4-(Furan-2-carbonyl)-piperazin-1-yl]-2-hydro...)
Affinity DataKi: >1.00E+3nMAssay Description:Beta-2 adrenergic receptor binding affinity by measuring the displacement of [3H]DHA binding in rat lung; Not Active means Ki >1000 nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Dog)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50086679(8-{3-[4-(4-Fluoro-phenyl)-piperazin-1-yl]-2-hydrox...)
Affinity DataKi: >1.00E+3nMAssay Description:Beta-2 adrenergic receptor binding affinity by measuring the displacement of [3H]DHA binding in rat lung; Not Active means Ki >1000 nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Dog)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50086662(4-{3-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-propyl}...)
Affinity DataKi: >1.00E+3nMAssay Description:Beta-2 adrenergic receptor binding affinity by measuring the displacement of [3H]DHA binding in rat lung; Not Active means Ki >1000 nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Dog)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50086678(7-{3-[4-(4-Fluoro-benzoyl)-piperazin-1-yl]-2-hydro...)
Affinity DataKi: >1.00E+3nMAssay Description:Beta-2 adrenergic receptor binding affinity by measuring the displacement of [3H]DHA binding in rat lung; Not Active means Ki >1000 nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Dog)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50086672(7-{3-[4-(Furan-2-carbonyl)-piperazin-1-yl]-2-hydro...)
Affinity DataKi: >1.00E+3nMAssay Description:Beta-2 adrenergic receptor binding affinity by measuring the displacement of [3H]DHA binding in rat lung; Not Active means Ki >1000 nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Dog)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50086668(7-{2-Hydroxy-3-[4-(2-methoxy-phenyl)-piperazin-1-y...)
Affinity DataKi: >1.00E+3nMAssay Description:Beta-2 adrenergic receptor binding affinity by measuring the displacement of [3H]DHA binding in rat lung; Not Active means Ki >1000 nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Dog)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50010841(CHEMBL98773 | 1-(4-Imidazol-1-yl-benzylamino)-3-o-...)
Affinity DataIC50: 1.20E+3nMAssay Description:Tested for Beta-2 adrenergic receptor selectivity in canine lung tissue in anesthetized dogsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2012
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Dog)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50064234(Dicyclopropyl-methanone O-(3-{2-[4-(3-dicyclopropy...)
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of beta-2 adrenergic receptor isolated from rat lung homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Dog)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50057128(A-80426 | (2-Benzofuran-6-yl-ethyl)-((R)-5-methoxy...)
Affinity DataKi:  1.74E+3nMAssay Description:Compound was evaluated for its binding affinity to beta-2 receptor in rat brain using [3H]- DHA radioligand assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/25/2012
Entry Details Article

TargetBeta-2 adrenergic receptor(Dog)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50064233(Dicyclopropyl-methanone O-{3-[2-(4-amino-phenyl)-1...)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of beta-2 adrenergic receptor isolated from rat lung homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Dog)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50001912(CHEMBL162513 | 4-Methanesulfonylamino-N-(4-phenyl-...)
Affinity DataIC50: 3.40E+3nMAssay Description:Binding affinity towards Beta-2 adrenergic receptor by displacing [3H]dihydroalprenolol, in partially purified membrane fractions from canine lung ti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Dog)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50001905(CHEMBL163587 | 4-Methanesulfonylamino-N-[4-(3-meth...)
Affinity DataIC50: 3.50E+3nMAssay Description:Binding affinity towards Beta-2 adrenergic receptor by displacing [3H]dihydroalprenolol, in partially purified membrane fractions from canine lung ti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Dog)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50087512((S)-adrenaline | (+)-adrenaline | CHEMBL42280)
Affinity DataKi:  3.70E+3nMAssay Description:Binding of [3H]dihydroalprenolol to beta-2 adrenergic receptor of rat cerebral cortical membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Dog)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50001914(CHEMBL350432 | N-[4-(3-Chloro-phenyl)-piperazin-2-...)
Affinity DataIC50: 3.80E+3nMAssay Description:Binding affinity towards Beta-2 adrenergic receptor by displacing [3H]dihydroalprenolol, in partially purified membrane fractions from canine lung ti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Dog)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50086677(6-{2-Hydroxy-3-[4-(2-methoxy-phenyl)-piperazin-1-y...)
Affinity DataKi:  4.00E+3nMAssay Description:Beta-2 adrenergic receptor binding affinity by measuring the displacement of [3H]DHA binding in rat lungMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Dog)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50001910(CHEMBL162200 | 4-(Methanesulfonyl-methyl-amino)-N-...)
Affinity DataIC50: 4.30E+3nMAssay Description:Binding affinity towards Beta-2 adrenergic receptor by displacing [3H]dihydroalprenolol, in partially purified membrane fractions from canine lung ti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Dog)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50001907(CHEMBL350847 | 4-Imidazol-1-yl-N-(4-phenyl-piperaz...)
Affinity DataIC50: 4.30E+3nMAssay Description:Binding affinity towards Beta-2 adrenergic receptor by displacing [3H]dihydroalprenolol, in partially purified membrane fractions from canine lung ti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Dog)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50010829(CHEMBL95966 | N-{4-[(2-Hydroxy-3-m-tolyloxy-propyl...)
Affinity DataIC50: 4.40E+3nMAssay Description:Tested for Beta-2 adrenergic receptor selectivity in canine lung tissue in anesthetized dogsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2012
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Dog)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50010837(CHEMBL95457 | 1-{2-[4-(3H-Imidazol-1-yl)-phenoxy]-...)
Affinity DataIC50: 4.50E+3nMAssay Description:Tested for Beta-2 adrenergic receptor selectivity in canine lung tissue in anesthetized dogsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2012
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Dog)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50001895(CHEMBL350581 | N-[4-(4-Phenyl-piperazin-2-ylmethox...)
Affinity DataIC50: 4.50E+3nMAssay Description:Binding affinity towards Beta-2 adrenergic receptor by displacing [3H]dihydroalprenolol, in partially purified membrane fractions from canine lung ti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Dog)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50001909(CHEMBL163153 | N-(4-{[(4-Phenyl-piperazin-2-ylmeth...)
Affinity DataIC50: 4.60E+3nMAssay Description:Binding affinity towards Beta-2 adrenergic receptor by displacing [3H]dihydroalprenolol, in partially purified membrane fractions from canine lung ti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Dog)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50086665(7-{3-[4-(4-Fluoro-phenyl)-piperazin-1-yl]-2-hydrox...)
Affinity DataKi:  4.80E+3nMAssay Description:Beta-2 adrenergic receptor binding affinity by measuring the displacement of [3H]DHA binding in rat lungMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Dog)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM25762(Sotalol,(-) | CHEMBL471 | cid_66245 | Sotalol,(+) ...)
Affinity DataIC50: 5.00E+3nMAssay Description:Binding affinity towards Beta-2 adrenergic receptor by displacing [3H]dihydroalprenolol, in partially purified membrane fractions from canine lung ti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Dog)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM25762(Sotalol,(-) | CHEMBL471 | cid_66245 | Sotalol,(+) ...)
Affinity DataIC50: 5.00E+3nMAssay Description:In vitro Beta-2 adrenergic receptor affinity in partially purified membrane fractions from canine lung tissue using [SH]dihydroalprenolol (4.5 nM)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
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