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Report error Found 665 for UniProtKB: P56481
TargetGastrin/cholecystokinin type B receptor(Mouse)
Ccipe-Faculte De Pharmacie

Curated by ChEMBL
LigandPNGBDBM50451028(PD-149164 | CHEMBL2062146)
Affinity DataIC50: 0.0830nMAssay Description:Binding affinity towards Cholecystokinin type B receptor in mouse cortex membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2012
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Mouse)
Ccipe-Faculte De Pharmacie

Curated by ChEMBL
LigandPNGBDBM50263229(CHEMBL505225 | CHEMBL505969 | 3-(4-(1-(2,3-dihydro...)
Affinity DataEC50:  0.140nMAssay Description:Agonist activity against mouse CCK1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Mouse)
Ccipe-Faculte De Pharmacie

Curated by ChEMBL
LigandPNGBDBM50062005(PD-135666 | 3-[2-(2-Adamantan-2-yl-acetylamino)-3-...)
Affinity DataKi:  0.148nMAssay Description:Cholecystokinin type B receptor binding assay performed on homogenized cerebral cortex from male mouseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2019
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Mouse)
Ccipe-Faculte De Pharmacie

Curated by ChEMBL
LigandPNGBDBM50062005(PD-135666 | 3-[2-(2-Adamantan-2-yl-acetylamino)-3-...)
Affinity DataIC50: 0.150nMAssay Description:Inhibitory concentration against radioligand [125I]Bolton-Hunter labeled CCK-8 to cholecystokinin type B receptor in the mouse cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Mouse)
Ccipe-Faculte De Pharmacie

Curated by ChEMBL
LigandPNGBDBM50062005(PD-135666 | 3-[2-(2-Adamantan-2-yl-acetylamino)-3-...)
Affinity DataIC50: 0.150nMAssay Description:Compound measured for half-maximal inhibition of specific binding of [125I]bolton Hunter CCK-26-33 to CCK-B receptor in the mouse cerebral cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetGastrin/cholecystokinin type B receptor(Mouse)
Ccipe-Faculte De Pharmacie

Curated by ChEMBL
LigandPNGBDBM50062005(PD-135666 | 3-[2-(2-Adamantan-2-yl-acetylamino)-3-...)
Affinity DataIC50: 0.150nMAssay Description:Half maximal inhibition of specific binding of [125I]Bolton-Hunter CCK-8 to Cholecystokinin type B receptor in the mouse cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2012
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Mouse)
Ccipe-Faculte De Pharmacie

Curated by ChEMBL
LigandPNGBDBM50062005(PD-135666 | 3-[2-(2-Adamantan-2-yl-acetylamino)-3-...)
Affinity DataIC50: 0.150nMAssay Description:Inhibition of [125I]CCK-8 to Cholecystokinin type B receptor in the mouse cerebral cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetGastrin/cholecystokinin type B receptor(Mouse)
Ccipe-Faculte De Pharmacie

Curated by ChEMBL
LigandPNGBDBM50073729((R)-3-[(S)-2-(Adamantan-2-yloxycarbonylamino)-3-(1...)
Affinity DataIC50: 0.150nMAssay Description:In vitro inhibition of [125I]- Bolton Hunter CCK-8 binding to Cholecystokinin type B receptor in the mouse cerebral cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

LigandPNGBDBM50016425(3-{2-[2-(2-{2-[2-(tert-Butoxycarbonyl-methyl-amino...)
Affinity DataKi:  0.191nMAssay Description:Binding affinity measured by inhibiting [3H]Boc[Nle28,31]CCK27-33 specific binding to Cholecystokinin receptor in mouse brain membranes at a KD conce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Mouse)
Ccipe-Faculte De Pharmacie

Curated by ChEMBL
LigandPNGBDBM50281737(PD-140376 | (R)-3-[(R)-2-(Adamantan-2-yloxycarbony...)
Affinity DataKi:  0.200nMAssay Description:The compound was evaluated for the inhibition of binding of [3H]-PD 140376 to Cholecystokinin type B receptor in mouse cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

TargetGastrin/cholecystokinin type B receptor(Mouse)
Ccipe-Faculte De Pharmacie

Curated by ChEMBL
LigandPNGBDBM50033586(3-[2-[(Adamantane-2-carbonyl)-amino]-3-(1H-indol-3...)
Affinity DataIC50: 0.210nMAssay Description:Inhibition of binding of [125I]Bolton-Hunter labeled CCK-8 to cholecystokinin type B receptor in the mouse cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2012
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Mouse)
Ccipe-Faculte De Pharmacie

Curated by ChEMBL
LigandPNGBDBM21147((3S)-3-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-[(3S)-3-...)
Affinity DataIC50: 0.300nMAssay Description:Half-maximal inhibition of specific binding of [125I]bolton hunter CCK-8 to mouse cerebral cortex Cholecystokinin type B receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2012
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Mouse)
Ccipe-Faculte De Pharmacie

Curated by ChEMBL
LigandPNGBDBM21147((3S)-3-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-[(3S)-3-...)
Affinity DataIC50: 0.300nMAssay Description:Inhibition of binding of [125I]Bolton-Hunter labeled CCK-8 to cholecystokinin type B receptor in the mouse cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2012
Entry Details Article
PubMed
LigandPNGBDBM21147((3S)-3-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-[(3S)-3-...)
Affinity DataKi:  0.300nMAssay Description:Potency in displacing [3H]propionyl-Cholecystokinin from mouse brain membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2019
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Mouse)
Ccipe-Faculte De Pharmacie

Curated by ChEMBL
LigandPNGBDBM21147((3S)-3-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-[(3S)-3-...)
Affinity DataIC50: 0.300nMAssay Description:Evaluated for inhibition of CCK-B receptor by displacing [125I]bolton hunter CCK-8 radioligand in the mouse cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Mouse)
Ccipe-Faculte De Pharmacie

Curated by ChEMBL
LigandPNGBDBM50033600(Asp-Tyr(SO3H)-Met-Gly-Trp-Met-Asp-Phe-NH2 | CHEMBL...)
Affinity DataIC50: 0.300nMAssay Description:Inhibition of binding of [125I]Bolton-Hunter labeled CCK-8 to cholecystokinin type B receptor in the mouse cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2012
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Mouse)
Ccipe-Faculte De Pharmacie

Curated by ChEMBL
LigandPNGBDBM21147((3S)-3-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-[(3S)-3-...)
Affinity DataIC50: 0.300nMAssay Description:Inhibition of [125I]- Bolton-Hunter CCK-26-33 binding to Cholecystokinin type B receptor of mouse cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

TargetGastrin/cholecystokinin type B receptor(Mouse)
Ccipe-Faculte De Pharmacie

Curated by ChEMBL
LigandPNGBDBM50245187(CHEMBL504861 | CHEMBL446789 | 3-(4-(1-(3-ethoxyphe...)
Affinity DataEC50:  0.300nMAssay Description:Agonist activity against mouse CCK1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Mouse)
Ccipe-Faculte De Pharmacie

Curated by ChEMBL
LigandPNGBDBM50281984((S)-3-[(Z)-2-(Adamantan-2-yloxycarbonylamino)-3-(1...)
Affinity DataIC50: 0.300nMAssay Description:Compound measured for half-maximal inhibition of specific binding of [125I]bolton Hunter CCK-26-33 to CCK-B receptor in the mouse cerebral cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetGastrin/cholecystokinin type B receptor(Mouse)
Ccipe-Faculte De Pharmacie

Curated by ChEMBL
LigandPNGBDBM21147((3S)-3-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-[(3S)-3-...)
Affinity DataIC50: 0.300nMAssay Description:Binding affinity towards Cholecystokinin type B receptor in mouse cortex membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2012
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Mouse)
Ccipe-Faculte De Pharmacie

Curated by ChEMBL
LigandPNGBDBM50281617(Asp Tyr (OSO3H) Met Gly Trp Met Asp Phe | CHEMBL26...)
Affinity DataIC50: 0.300nMAssay Description:Compound was tested for the inhibition of specific binding of [125I]bolton Hunter CCK-8 to Cholecystokinin type B receptor in mouse cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetGastrin/cholecystokinin type B receptor(Mouse)
Ccipe-Faculte De Pharmacie

Curated by ChEMBL
LigandPNGBDBM50456331(CHEMBL2111203)
Affinity DataIC50: 0.340nMAssay Description:Inhibition of binding of [125I]Bolton-Hunter labeled CCK-8 to cholecystokinin type B receptor in the mouse cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2012
Entry Details Article
PubMed
LigandPNGBDBM21147((3S)-3-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-[(3S)-3-...)
Affinity DataKi:  0.491nMAssay Description:Binding affinity measured by inhibiting [3H]Boc[Nle28,31]CCK27-33 specific binding to Cholecystokinin receptor in mouse brain membranes at a KD conce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Mouse)
Ccipe-Faculte De Pharmacie

Curated by ChEMBL
LigandPNGBDBM50456329(CHEMBL2111261)
Affinity DataIC50: 0.510nMAssay Description:Inhibition of binding of [125I]Bolton-Hunter labeled CCK-8 to cholecystokinin type B receptor in the mouse cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2012
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Mouse)
Ccipe-Faculte De Pharmacie

Curated by ChEMBL
LigandPNGBDBM50230677(CHEMBL3351022)
Affinity DataKi:  0.513nMAssay Description:Cholecystokinin type B receptor binding assay performed on homogenized cerebral cortex from male mouseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2019
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Mouse)
Ccipe-Faculte De Pharmacie

Curated by ChEMBL
LigandPNGBDBM50285623((R)-3-[(R)-2-(Adamantan-2-yloxycarbonylamino)-3-(1...)
Affinity DataKi:  0.520nMAssay Description:Binding affinity towards CCK-B receptor in mouse cerebral cortex membrane using [125I]bolton assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/26/2012
Entry Details Article

TargetGastrin/cholecystokinin type B receptor(Mouse)
Ccipe-Faculte De Pharmacie

Curated by ChEMBL
LigandPNGBDBM50033587([1-(1-Hydroxymethyl-2-phenyl-ethylcarbamoyl)-2-(1H...)
Affinity DataIC50: 0.600nMAssay Description:Inhibition of binding of [125I]Bolton-Hunter labeled CCK-8 to cholecystokinin type B receptor in the mouse cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2012
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Mouse)
Ccipe-Faculte De Pharmacie

Curated by ChEMBL
LigandPNGBDBM50007439(CHEMBL341460 | 3-{2-[2-(Adamantan-2-yloxycarbonyla...)
Affinity DataIC50: 0.700nMAssay Description:Half-maximal inhibition of specific binding of [125I]bolton hunter CCK-8 to mouse cerebral cortex Cholecystokinin type B receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2012
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Mouse)
Ccipe-Faculte De Pharmacie

Curated by ChEMBL
LigandPNGBDBM50033606(3-{2-[2-[(Adamantane-2-carbonyl)-amino]-3-(1H-indo...)
Affinity DataIC50: 0.700nMAssay Description:Inhibition of binding of [125I]Bolton-Hunter labeled CCK-8 to cholecystokinin type B receptor in the mouse cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2012
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Mouse)
Ccipe-Faculte De Pharmacie

Curated by ChEMBL
LigandPNGBDBM50230683(CHEMBL3351024)
Affinity DataKi:  0.708nMAssay Description:Cholecystokinin type B receptor binding assay performed on homogenized cerebral cortex from male mouseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2019
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Mouse)
Ccipe-Faculte De Pharmacie

Curated by ChEMBL
LigandPNGBDBM50471066(CHEMBL415936)
Affinity DataKi:  0.741nMAssay Description:In vitro inhibitory activity against Cholecystokinin type B receptor using [125I]BH-CCK-8S as radioligand in mouse cortical membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Mouse)
Ccipe-Faculte De Pharmacie

Curated by ChEMBL
LigandPNGBDBM50263231(sodium 3-(4-(1-(3-ethoxyphenyl)-2-p-tolyl-1H-imida...)
Affinity DataEC50:  0.780nMAssay Description:Agonist activity against mouse CCK1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Mouse)
Ccipe-Faculte De Pharmacie

Curated by ChEMBL
LigandPNGBDBM50033604(3-{2-[2-[(Adamantane-2-carbonyl)-amino]-3-(1H-indo...)
Affinity DataIC50: 0.800nMAssay Description:Inhibition of binding of [125I]Bolton-Hunter labeled CCK-8 to cholecystokinin type B receptor in the mouse cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2012
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Mouse)
Ccipe-Faculte De Pharmacie

Curated by ChEMBL
LigandPNGBDBM50024321(CHEMBL1328 | Peptavlon | ICI-50123 | 3-{2-[2-(3-te...)
Affinity DataIC50: 0.800nMAssay Description:Half-maximal inhibition of specific binding of [125I]bolton hunter CCK-8 to mouse cerebral cortex Cholecystokinin type B receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2012
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Mouse)
Ccipe-Faculte De Pharmacie

Curated by ChEMBL
LigandPNGBDBM50452998(CHEMBL2112693)
Affinity DataIC50: 0.800nMAssay Description:Half-maximal inhibition of specific binding of [125I]bolton hunter CCK-8 to mouse cerebral cortex Cholecystokinin type B receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2012
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Mouse)
Ccipe-Faculte De Pharmacie

Curated by ChEMBL
LigandPNGBDBM50024321(CHEMBL1328 | Peptavlon | ICI-50123 | 3-{2-[2-(3-te...)
Affinity DataIC50: 0.800nMAssay Description:Inhibition of binding of [125I]Bolton-Hunter labeled CCK-8 to cholecystokinin type B receptor in the mouse cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2012
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Mouse)
Ccipe-Faculte De Pharmacie

Curated by ChEMBL
LigandPNGBDBM50024321(CHEMBL1328 | Peptavlon | ICI-50123 | 3-{2-[2-(3-te...)
Affinity DataIC50: 0.800nMAssay Description:Evaluated for inhibition of CCK-B receptor by displacing [125I]bolton hunter CCK-8 radioligand in the mouse cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Mouse)
Ccipe-Faculte De Pharmacie

Curated by ChEMBL
LigandPNGBDBM50007449(CHEMBL337384 | 3-{2-[2-(Adamantan-2-yloxycarbonyla...)
Affinity DataIC50: 0.800nMAssay Description:Half-maximal inhibition of specific binding of [125I]bolton hunter CCK-8 to mouse cerebral cortex Cholecystokinin type B receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2012
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Mouse)
Ccipe-Faculte De Pharmacie

Curated by ChEMBL
LigandPNGBDBM50285625(PD-142251 | (R)-3-[2-((R)-Adamantan-2-yloxycarbony...)
Affinity DataKi:  0.880nMAssay Description:Binding affinity towards CCK-B receptor in mouse cerebral cortex membrane using [125I]bolton assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/26/2012
Entry Details Article

TargetGastrin/cholecystokinin type B receptor(Mouse)
Ccipe-Faculte De Pharmacie

Curated by ChEMBL
LigandPNGBDBM50062000(2-[(R)-2-(Adamantan-2-yloxycarbonylamino)-3-(1H-in...)
Affinity DataIC50: 0.990nMAssay Description:Inhibitory concentration against radioligand [125I]Bolton-Hunter labeled CCK-8 to cholecystokinin type B receptor in the mouse cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Mouse)
Ccipe-Faculte De Pharmacie

Curated by ChEMBL
LigandPNGBDBM50063665(N-(3-nitrophenyl)-2-[3,4-dihydro-3-[3-(1-methyleth...)
Affinity DataIC50: 1nMAssay Description:Binding affinity towards Cholecystokinin type B receptor (CCK-B) receptor in mouse cerebral cortex using [125I]bolton Hunter CCK-8 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Mouse)
Ccipe-Faculte De Pharmacie

Curated by ChEMBL
LigandPNGBDBM50213845(CHEMBL14557)
Affinity DataKi:  1nMAssay Description:Inhibition of 20 pM [125I]BH-CCK-8S binding to mouse cortical membrane Cholecystokinin 2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Mouse)
Ccipe-Faculte De Pharmacie

Curated by ChEMBL
LigandPNGBDBM50230676(CHEMBL3351013)
Affinity DataKi:  1.10nMAssay Description:Cholecystokinin type B receptor binding assay performed on homogenized cerebral cortex from male mouseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2019
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Mouse)
Ccipe-Faculte De Pharmacie

Curated by ChEMBL
LigandPNGBDBM50213845(CHEMBL14557)
Affinity DataKi:  1.10nMAssay Description:In vitro inhibitory activity against Cholecystokinin type B receptor using [125I]BH-CCK-8S as radioligand in mouse cortical membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Mouse)
Ccipe-Faculte De Pharmacie

Curated by ChEMBL
LigandPNGBDBM50213845(CHEMBL14557)
Affinity DataKi:  1.10nMAssay Description:Displacement of binding of [125I]CCK-8S to Cholecystokinin type B receptor in mouse cerebral cortex homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Mouse)
Ccipe-Faculte De Pharmacie

Curated by ChEMBL
LigandPNGBDBM50471075(CHEMBL299540)
Affinity DataKi:  1.20nMAssay Description:In vitro inhibitory activity against Cholecystokinin type B receptor using [125I]BH-CCK-8S as radioligand in mouse cortical membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Mouse)
Ccipe-Faculte De Pharmacie

Curated by ChEMBL
LigandPNGBDBM50033592(3-{2-[3-(1H-Indol-3-yl)-2-methyl-2-(2-methyl-cyclo...)
Affinity DataIC50: 1.20nMAssay Description:Inhibition of binding of [125I]Bolton-Hunter labeled CCK-8 to cholecystokinin type B receptor in the mouse cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2012
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Mouse)
Ccipe-Faculte De Pharmacie

Curated by ChEMBL
LigandPNGBDBM50471067(CHEMBL298521)
Affinity DataKi:  1.20nMAssay Description:In vitro inhibitory activity against Cholecystokinin type B receptor using [125I]BH-CCK-8S as radioligand in mouse cortical membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Mouse)
Ccipe-Faculte De Pharmacie

Curated by ChEMBL
LigandPNGBDBM50063640(N-(3-cyanobenzene)-2-[3,4-dihydro-3-[3-(1-methylet...)
Affinity DataIC50: 1.20nMAssay Description:Binding affinity towards Cholecystokinin type B receptor (CCK-B) receptor in mouse cerebral cortex using [125I]bolton Hunter CCK-8 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Mouse)
Ccipe-Faculte De Pharmacie

Curated by ChEMBL
LigandPNGBDBM21147((3S)-3-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-[(3S)-3-...)
Affinity DataIC50: 1.30nMAssay Description:In vitro binding affinity against Cholecystokinin type B receptor in mouse cerebral cortical membranes using [125I]Tyr(SO3H)27]-CCK-8 binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
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