Compile Data Set for Download or QSAR
Report error Found 29 for UniProtKB: Q01063
LigandChemical structure of BindingDB Monomer ID 50470788BDBM50470788(CHEMBL278386)
Affinity DataIC50: 3nMAssay Description:Displacement of [3H]rolipram from mouse brain homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50470784BDBM50470784(CHEMBL282934)
Affinity DataIC50: 3nMAssay Description:Displacement of [3H]rolipram from mouse brain homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 14361BDBM14361(Adeo | 4-(3-cyclopentyloxy-4-methoxy-phenyl)pyrrol...)
Affinity DataIC50: 4nMAssay Description:Inhibition of [3H]rolipram binding to Phosphodiesterase 4 (PDE IV)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2018
Entry Details
PDB3D3D Structure (crystal)
LigandChemical structure of BindingDB Monomer ID 14361BDBM14361(Adeo | 4-(3-cyclopentyloxy-4-methoxy-phenyl)pyrrol...)
Affinity DataIC50: 4nMAssay Description:Displacement of [3H]rolipram from mouse brain homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
LigandChemical structure of BindingDB Monomer ID 14361BDBM14361(Adeo | 4-(3-cyclopentyloxy-4-methoxy-phenyl)pyrrol...)
Affinity DataIC50: 4nMAssay Description:Displacement of [3H]-Rolipram from mouse brain homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2018
Entry Details
PDB3D3D Structure (crystal)
LigandChemical structure of BindingDB Monomer ID 50470782BDBM50470782(CHEMBL280185)
Affinity DataIC50: 5nMAssay Description:Displacement of [3H]rolipram from mouse brain homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50470786BDBM50470786(CHEMBL21964)
Affinity DataIC50: 9nMAssay Description:Displacement of [3H]rolipram from mouse brain homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50470779BDBM50470779(CHEMBL21463)
Affinity DataIC50: 15nMAssay Description:Displacement of [3H]rolipram from mouse brain homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50470781BDBM50470781(CHEMBL281781)
Affinity DataIC50: 15nMAssay Description:Displacement of [3H]rolipram from mouse brain homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50213340BDBM50213340(CHEMBL58915)
Affinity DataIC50: 32nMAssay Description:Displacement of [3H]-Rolipram from mouse brain homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2018
Entry Details

LigandChemical structure of BindingDB Monomer ID 50213338BDBM50213338(CHEMBL294883)
Affinity DataIC50: 78nMAssay Description:Displacement of [3H]-Rolipram from mouse brain homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2018
Entry Details

LigandChemical structure of BindingDB Monomer ID 50470778BDBM50470778(CHEMBL21839)
Affinity DataIC50: 111nMAssay Description:Displacement of [3H]rolipram from mouse brain homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50470780BDBM50470780(CHEMBL21305)
Affinity DataIC50: 129nMAssay Description:Displacement of [3H]rolipram from mouse brain homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50457395BDBM50457395(CHEMBL4209111 | US11401286, Example 220)
Affinity DataIC50: 130nMAssay Description:Allosteric modulation of mouse PDE4DMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50470783BDBM50470783(CHEMBL21327)
Affinity DataIC50: 130nMAssay Description:Displacement of [3H]rolipram from mouse brain homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50213341BDBM50213341(CHEMBL59269)
Affinity DataIC50: 130nMAssay Description:Displacement of [3H]-Rolipram from mouse brain homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2018
Entry Details

LigandChemical structure of BindingDB Monomer ID 50213339BDBM50213339(CHEMBL291537)
Affinity DataIC50: 220nMAssay Description:Displacement of [3H]-Rolipram from mouse brain homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2018
Entry Details

LigandChemical structure of BindingDB Monomer ID 50470785BDBM50470785(CHEMBL422219)
Affinity DataIC50: 323nMAssay Description:Displacement of [3H]rolipram from mouse brain homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50470776BDBM50470776(CHEMBL280729)
Affinity DataIC50: 653nMAssay Description:Displacement of [3H]rolipram from mouse brain homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50470787BDBM50470787(CHEMBL22461)
Affinity DataIC50: 1.68E+3nMAssay Description:Displacement of [3H]rolipram from mouse brain homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50470775BDBM50470775(CHEMBL22898)
Affinity DataIC50: 1.90E+3nMAssay Description:Displacement of [3H]rolipram from mouse brain homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50213335BDBM50213335(CHEMBL60985)
Affinity DataIC50: 3.20E+3nMAssay Description:Inhibition of [3H]rolipram binding to Phosphodiesterase 4 (PDE IV)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2018
Entry Details

LigandChemical structure of BindingDB Monomer ID 50213299BDBM50213299(CHEMBL291838)
Affinity DataIC50: 4.60E+3nMAssay Description:Inhibition of [3H]rolipram binding to Phosphodiesterase 4 (PDE IV)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2018
Entry Details

LigandChemical structure of BindingDB Monomer ID 50213337BDBM50213337(CHEMBL60073)
Affinity DataIC50: 5.91E+3nMAssay Description:Displacement of [3H]-Rolipram from mouse brain homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2018
Entry Details

LigandChemical structure of BindingDB Monomer ID 50213301BDBM50213301(CHEMBL61884)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of [3H]rolipram binding to Phosphodiesterase 4 (PDE IV)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2018
Entry Details

LigandChemical structure of BindingDB Monomer ID 50213300BDBM50213300(CHEMBL294606)
Affinity DataIC50: 5.70E+4nMAssay Description:Inhibition of [3H]rolipram binding to Phosphodiesterase 4 (PDE IV)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2018
Entry Details

LigandChemical structure of BindingDB Monomer ID 50213336BDBM50213336(CHEMBL60007)
Affinity DataIC50: 5.80E+4nMAssay Description:Inhibition of [3H]rolipram binding to Phosphodiesterase 4 (PDE IV)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2018
Entry Details

LigandChemical structure of BindingDB Monomer ID 50213298BDBM50213298(CHEMBL59408)
Affinity DataIC50: 6.20E+4nMAssay Description:Inhibition of [3H]rolipram binding to Phosphodiesterase 4 (PDE IV)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2018
Entry Details

LigandChemical structure of BindingDB Monomer ID 50213302BDBM50213302(CHEMBL60060)
Affinity DataIC50: 6.60E+4nMAssay Description:Inhibition of [3H]rolipram binding to Phosphodiesterase 4 (PDE IV)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2018
Entry Details