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Target5-hydroxytryptamine receptor 4(Human)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM85027(1-(7-Chloro-8-amino-1,4-benzodioxane-5-yl)-3-[1-[3...)
Affinity DataKi:  0.000580nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/1/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Human)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM85027(1-(7-Chloro-8-amino-1,4-benzodioxane-5-yl)-3-[1-[3...)
Affinity DataKi:  0.000630nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/1/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Human)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM85020(GR-125487 | 5-Fluoro-2-methoxy-1H-indole-3-carboxy...)
Affinity DataKi:  0.000870nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/1/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Human)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM50483188(CHEMBL1632166)
Affinity DataKi:  0.00145nMAssay Description:Displacement of [3H]GR113808 from human 5HT4 receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Human)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM198005(US9221790, 15)
Affinity DataIC50: 0.00200nMAssay Description:The binding affinity of the compounds for a human 5-HT4 receptor was assayed according to the method as disclosed in the literature [Wyngaert et al.,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2016
Entry Details
US Patent

Target5-hydroxytryptamine receptor 4(Human)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM197995(US9221790, 5)
Affinity DataIC50: 0.00500nMAssay Description:The binding affinity of the compounds for a human 5-HT4 receptor was assayed according to the method as disclosed in the literature [Wyngaert et al.,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2016
Entry Details
US Patent

Target5-hydroxytryptamine receptor 4(Human)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM85026(SB-207266 | N-(1-Butylpiperidine-4-ylmethyl)-1,2-(...)
Affinity DataKi:  0.0100nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/1/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Human)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM29525(GR 113808 | [3H] GR 113808 | CHEMBL518682 | 3H-GR1...)
Affinity DataKi:  0.0200nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/1/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Human)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM85020(GR-125487 | 5-Fluoro-2-methoxy-1H-indole-3-carboxy...)
Affinity DataKi:  0.0200nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/1/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Human)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM82505(CAS_121881 | NSC_121881 | SB204070)
Affinity DataKi:  0.0300nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Human)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM197993(US9221790, 3)
Affinity DataIC50: 0.0390nMAssay Description:The binding affinity of the compounds for a human 5-HT4 receptor was assayed according to the method as disclosed in the literature [Wyngaert et al.,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2016
Entry Details
US Patent

Target5-hydroxytryptamine receptor 4(Human)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM50399614(CHEMBL2181170)
Affinity DataKi:  0.0398nMAssay Description:Displacement of radioligand from human 5HT4R by Cerep protocol based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Human)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM29525(GR 113808 | [3H] GR 113808 | CHEMBL518682 | 3H-GR1...)
Affinity DataKi:  0.0398nMAssay Description:Displacement of [3H]GR113808 from human 5-HT4B receptor expressed in HEK293 cells after 1 hr by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Human)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM50399614(CHEMBL2181170)
Affinity DataKi:  0.0400nMAssay Description:Displacement of radioligand from human 5HT4R by Cerep protocol based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Human)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM50483175(CHEMBL1632165)
Affinity DataKi:  0.0427nMAssay Description:Displacement of [3H]GR113808 from human 5HT4 receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Human)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM29525(GR 113808 | [3H] GR 113808 | CHEMBL518682 | 3H-GR1...)
Affinity DataKi:  0.0500nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/30/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Human)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM29525(GR 113808 | [3H] GR 113808 | CHEMBL518682 | 3H-GR1...)
Affinity DataKi:  0.0500nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/30/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Human)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM50327858(CHEMBL114112 | SB207710 | 8-Amino-7-iodo-2,3-dihyd...)
Affinity DataKi:  0.0500nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/30/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Human)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM50023377(CHEMBL3329805)
Affinity DataKi:  0.0501nMAssay Description:Displacement of [3H]GR113808 from human 5HT4b receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Human)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM85026(SB-207266 | N-(1-Butylpiperidine-4-ylmethyl)-1,2-(...)
Affinity DataKi:  0.0525nMAssay Description:Displacement of [3H]GR113808 from human 5HT4 receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Human)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM50483174(CHEMBL1632163)
Affinity DataKi:  0.0537nMAssay Description:Displacement of [3H]GR113808 from human 5HT4 receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Human)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM82505(CAS_121881 | NSC_121881 | SB204070)
Affinity DataKi:  0.0600nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Human)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM50483187(CHEMBL1632169)
Affinity DataKi:  0.0646nMAssay Description:Displacement of [3H]GR113808 from human 5HT4 receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Human)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM197997(US9221790, 7)
Affinity DataIC50: 0.0670nMAssay Description:The binding affinity of the compounds for a human 5-HT4 receptor was assayed according to the method as disclosed in the literature [Wyngaert et al.,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2016
Entry Details
US Patent

Target5-hydroxytryptamine receptor 4(Human)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM29525(GR 113808 | [3H] GR 113808 | CHEMBL518682 | 3H-GR1...)
Affinity DataKi:  0.0700nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Human)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM29525(GR 113808 | [3H] GR 113808 | CHEMBL518682 | 3H-GR1...)
Affinity DataKi:  0.0741nMAssay Description:Antagonistic activity at human 5HT4 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Human)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM198000(US9221790, 10)
Affinity DataIC50: 0.0760nMAssay Description:The binding affinity of the compounds for a human 5-HT4 receptor was assayed according to the method as disclosed in the literature [Wyngaert et al.,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2016
Entry Details
US Patent

Target5-hydroxytryptamine receptor 4(Human)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM29525(GR 113808 | [3H] GR 113808 | CHEMBL518682 | 3H-GR1...)
Affinity DataKi:  0.0780nMAssay Description:Binding affinity was determined against cloned 5-hydroxytryptamine 4D receptor isoform expressed in COS-7 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Human)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM29525(GR 113808 | [3H] GR 113808 | CHEMBL518682 | 3H-GR1...)
Affinity DataKi:  0.0790nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/30/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Human)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM50327858(CHEMBL114112 | SB207710 | 8-Amino-7-iodo-2,3-dihyd...)
Affinity DataKi:  0.0790nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/30/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Human)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM50398985(CHEMBL2177130)
Affinity DataKi:  0.0794nMAssay Description:Displacement of [3H](1-(2-(methylsulfonamido)ethyl)piperidin-4-yl)methyl 1-methyl-1H-indole-3-carboxylate from human 5HT4R expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Human)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM50023365(CHEMBL3329814)
Affinity DataKi:  0.0794nMAssay Description:Displacement of [3H]GR113808 from human 5HT4b receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Human)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM29525(GR 113808 | [3H] GR 113808 | CHEMBL518682 | 3H-GR1...)
Affinity DataKi:  0.0900nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/1/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Human)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM85026(SB-207266 | N-(1-Butylpiperidine-4-ylmethyl)-1,2-(...)
Affinity DataKi:  0.100nMAssay Description:Displacement of [3H]GR113808 from human 5-HT4B receptor expressed in HEK293 cells after 1 hr by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Human)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM82505(CAS_121881 | NSC_121881 | SB204070)
Affinity DataKi:  0.100nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Human)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM50398983(CHEMBL2179697)
Affinity DataKi:  0.100nMAssay Description:Displacement of [3H](1-(2-(methylsulfonamido)ethyl)piperidin-4-yl)methyl 1-methyl-1H-indole-3-carboxylate from human 5HT4R expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Human)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM50456128(CHEMBL4215329)
Affinity DataEC50:  0.100nMAssay Description:Agonist activity at recombinant human 5-HT4E receptor expressed in CHO cells assessed as induction of c-AMP accumulation after 4 hrs by luciferase re...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Human)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM29525(GR 113808 | [3H] GR 113808 | CHEMBL518682 | 3H-GR1...)
Affinity DataKi:  0.100nMAssay Description:Binding affinity was determined against cloned 5-hydroxytryptamine 4E receptor isoform expressed in C6 glial cells incubated with 0.2 nM [3H]GR-11380...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Human)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM82505(CAS_121881 | NSC_121881 | SB204070)
Affinity DataKi:  0.100nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/1/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Human)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM50483173(CHEMBL1632157)
Affinity DataKi:  0.102nMAssay Description:Displacement of [3H]GR113808 from human 5HT4 receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Human)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM197996(US9221790, 6)
Affinity DataIC50: 0.103nMAssay Description:The binding affinity of the compounds for a human 5-HT4 receptor was assayed according to the method as disclosed in the literature [Wyngaert et al.,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2016
Entry Details
US Patent

Target5-hydroxytryptamine receptor 4(Human)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM50483172(CHEMBL1632158)
Affinity DataKi:  0.107nMAssay Description:Displacement of [3H]GR113808 from human 5HT4 receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Human)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM50492064(CHEMBL2391994)
Affinity DataKi:  0.126nMAssay Description:Displacement of [3H]GR113808 from human 5-HT4B receptor expressed in HEK293 cells after 1 hr by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Human)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM198003(US9221790, 13)
Affinity DataIC50: 0.134nMAssay Description:The binding affinity of the compounds for a human 5-HT4 receptor was assayed according to the method as disclosed in the literature [Wyngaert et al.,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2016
Entry Details
US Patent

Target5-hydroxytryptamine receptor 4(Human)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM50483186(CHEMBL1632167)
Affinity DataKi:  0.141nMAssay Description:Displacement of [3H]GR113808 from human 5HT4 receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Human)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM29525(GR 113808 | [3H] GR 113808 | CHEMBL518682 | 3H-GR1...)
Affinity DataKi:  0.150nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Human)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM29525(GR 113808 | [3H] GR 113808 | CHEMBL518682 | 3H-GR1...)
Affinity DataKi:  0.150nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/1/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Human)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM50398598(CHEMBL2152922)
Affinity DataKi:  0.150nMAssay Description:Displacement of [3H]GR113808 from human 5HT4D receptor expressed in HEK293 cells after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Human)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM85020(GR-125487 | 5-Fluoro-2-methoxy-1H-indole-3-carboxy...)
Affinity DataKi:  0.150nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/1/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Human)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM50398981(CHEMBL2179699)
Affinity DataKi:  0.158nMAssay Description:Displacement of [3H](1-(2-(methylsulfonamido)ethyl)piperidin-4-yl)methyl 1-methyl-1H-indole-3-carboxylate from human 5HT4R expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
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