Compile Data Set for Download or QSAR
Report error Found 16 of affinity data for UniProtKB/TrEMBL: Q59514
TargetBeta-lactamase BRO-1(Moraxella catarrhalis)TBA
LigandChemical structure of BindingDB Monomer ID 50212637BDBM50212637(CHEMBL72046)
Affinity DataIC50: 2.85nMAssay Description:Inhibitory activity against Branhamella catarrhalis 89001 Class-III BRO-1 type beta-lactamase enzymeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2018
Entry Details

TargetBeta-lactamase BRO-1(Moraxella catarrhalis)TBA
LigandChemical structure of BindingDB Monomer ID 50212640BDBM50212640(CHEMBL423309)
Affinity DataIC50: 2.89nMAssay Description:Inhibitory activity against Branhamella catarrhalis 89001 Class-III BRO-1 type beta-lactamase enzymeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2018
Entry Details

TargetBeta-lactamase BRO-1(Moraxella catarrhalis)TBA
LigandChemical structure of BindingDB Monomer ID 50212639BDBM50212639(CHEMBL302241)
Affinity DataIC50: 2.90nMAssay Description:Inhibitory activity against Branhamella catarrhalis 89001 Class-III BRO-1 type beta-lactamase enzymeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2018
Entry Details

TargetBeta-lactamase BRO-1(Moraxella catarrhalis)TBA
LigandChemical structure of BindingDB Monomer ID 50212634BDBM50212634(CHEMBL309009)
Affinity DataIC50: 5.23nMAssay Description:Inhibitory activity against Branhamella catarrhalis 89001 Class-III BRO-1 type beta-lactamase enzymeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2018
Entry Details

TargetBeta-lactamase BRO-1(Moraxella catarrhalis)TBA
LigandChemical structure of BindingDB Monomer ID 50212638BDBM50212638(CHEMBL302512)
Affinity DataIC50: 8.64nMAssay Description:Inhibitory activity against Branhamella catarrhalis 89001 Class-III BRO-1 type beta-lactamase enzymeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2018
Entry Details

TargetBeta-lactamase BRO-1(Moraxella catarrhalis)TBA
LigandChemical structure of BindingDB Monomer ID 50212641BDBM50212641(Brobactam)
Affinity DataIC50: 10.7nMAssay Description:Inhibitory activity against Branhamella catarrhalis 89001 Class-III BRO-1 type beta-lactamase enzymeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2018
Entry Details

TargetBeta-lactamase BRO-1(Moraxella catarrhalis)TBA
LigandChemical structure of BindingDB Monomer ID 50212646BDBM50212646(CHEMBL72972)
Affinity DataIC50: 13.1nMAssay Description:Inhibitory activity against Branhamella catarrhalis 89001 Class-III BRO-1 type beta-lactamase enzymeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2018
Entry Details

TargetBeta-lactamase BRO-1(Moraxella catarrhalis)TBA
LigandChemical structure of BindingDB Monomer ID 50212642BDBM50212642(CHEMBL70269)
Affinity DataIC50: 23.3nMAssay Description:Inhibitory activity against Branhamella catarrhalis 89001 Class-III BRO-1 type beta-lactamase enzymeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2018
Entry Details

TargetBeta-lactamase BRO-1(Moraxella catarrhalis)TBA
LigandChemical structure of BindingDB Monomer ID 50021959BDBM50021959(antibiotic MM 14151 | CHEMBL777 | MM 14151 | clavu...)
Affinity DataIC50: 30.1nMAssay Description:Inhibitory activity against Branhamella catarrhalis 89001 Class-III BRO-1 type beta-lactamase enzymeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2018
Entry Details

TargetBeta-lactamase BRO-1(Moraxella catarrhalis)TBA
LigandChemical structure of BindingDB Monomer ID 50053173BDBM50053173((2S,3S,5R)-3-Methyl-4,4,7-trioxo-3-[1,2,3]triazol-...)
Affinity DataIC50: 33.3nMAssay Description:Inhibitory activity against Branhamella catarrhalis 89001 Class-III BRO-1 type beta-lactamase enzymeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2018
Entry Details

TargetBeta-lactamase BRO-1(Moraxella catarrhalis)TBA
LigandChemical structure of BindingDB Monomer ID 50212635BDBM50212635(CHEMBL415266)
Affinity DataIC50: 50.7nMAssay Description:Inhibitory activity against Branhamella catarrhalis 89001 Class-III BRO-1 type beta-lactamase enzymeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2018
Entry Details

TargetBeta-lactamase BRO-1(Moraxella catarrhalis)TBA
LigandChemical structure of BindingDB Monomer ID 50212643BDBM50212643(CHEMBL308516)
Affinity DataIC50: 56.1nMAssay Description:Inhibitory activity against Branhamella catarrhalis 89001 Class-III BRO-1 type beta-lactamase enzymeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2018
Entry Details

TargetBeta-lactamase BRO-1(Moraxella catarrhalis)TBA
LigandChemical structure of BindingDB Monomer ID 50212644BDBM50212644(CHEMBL73450)
Affinity DataIC50: 63.7nMAssay Description:Inhibitory activity against Branhamella catarrhalis 89001 Class-III BRO-1 type beta-lactamase enzymeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2018
Entry Details

TargetBeta-lactamase BRO-1(Moraxella catarrhalis)TBA
LigandChemical structure of BindingDB Monomer ID 50212645BDBM50212645(CHEMBL305908)
Affinity DataIC50: 65.9nMAssay Description:Inhibitory activity against Branhamella catarrhalis 89001 Class-III BRO-1 type beta-lactamase enzymeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2018
Entry Details

TargetBeta-lactamase BRO-1(Moraxella catarrhalis)TBA
LigandChemical structure of BindingDB Monomer ID 50212636BDBM50212636(CHEMBL310221)
Affinity DataIC50: 80.5nMAssay Description:Inhibitory activity against Branhamella catarrhalis 89001 Class-III BRO-1 type beta-lactamase enzymeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2018
Entry Details

TargetBeta-lactamase BRO-1(Moraxella catarrhalis)TBA
LigandChemical structure of BindingDB Monomer ID 50021954BDBM50021954(UNASYN | 3,3-Dimethyl-4,4,7-trioxo-4lambda*6*-thia...)
Affinity DataIC50: 107nMAssay Description:Inhibitory activity against Branhamella catarrhalis 89001 Class-III BRO-1 type beta-lactamase enzymeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2018
Entry Details