Compile Data Set for Download or QSAR
Report error Found 37 of affinity data for UniProtKB/TrEMBL: Q5QD14
TargetTrace amine-associated receptor 5(Mouse)
University of Genoa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50227979BDBM50227979(CHEMBL4084561)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at mouse TAAR5 expressed in HEK293 cells assessed as cAMP accumulation after 20 mins by BRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2019
Entry Details Article
PubMed
TargetTrace amine-associated receptor 5(Mouse)
University of Genoa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50227829BDBM50227829(CHEBI:8455 | Proguanil | CHLOROGUANIDE)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at mouse TAAR5 expressed in HEK293 cells assessed as cAMP accumulation after 20 mins by BRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2019
Entry Details Article
PubMed
TargetTrace amine-associated receptor 5(Mouse)
University of Genoa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50227826BDBM50227826(CHEMBL4069147)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at mouse TAAR5 expressed in HEK293 cells assessed as cAMP accumulation after 20 mins by BRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2019
Entry Details Article
PubMed
TargetTrace amine-associated receptor 5(Mouse)
University of Genoa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 18512BDBM18512(cid_4993 | CHEMBL36 | 5-(4-chlorophenyl)-6-ethylpy...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at mouse TAAR5 expressed in HEK293 cells assessed as cAMP accumulation after 20 mins by BRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2019
Entry Details Article
PubMed
TargetTrace amine-associated receptor 5(Mouse)
University of Genoa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50053615BDBM50053615(m-chlorophenylbiguanidine | 3-Chloro-Phenyl biguan...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at mouse TAAR5 expressed in HEK293 cells assessed as cAMP accumulation after 20 mins by BRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2019
Entry Details Article
PubMed
TargetTrace amine-associated receptor 5(Mouse)
University of Genoa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50053629BDBM50053629(2-Chloro-Phenyl biguanide | N-(2-chlorophenyl)imid...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at mouse TAAR5 expressed in HEK293 cells assessed as cAMP accumulation after 20 mins by BRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2019
Entry Details Article
PubMed
TargetTrace amine-associated receptor 5(Mouse)
University of Genoa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50293273BDBM50293273(CHEMBL4172220)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at mouse TAAR5 expressed in HEK293 cells assessed as cAMP accumulation after 20 mins by BRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/5/2020
Entry Details Article
PubMed
TargetTrace amine-associated receptor 5(Mouse)
University of Genoa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50227830BDBM50227830(CHEMBL4099661)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at mouse TAAR5 expressed in HEK293 cells assessed as cAMP accumulation after 20 mins by BRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2019
Entry Details Article
PubMed
TargetTrace amine-associated receptor 5(Mouse)
University of Genoa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50100977BDBM50100977(N-(3,4-dichlorophenyl)imidodicarbonimidic diamide ...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at mouse TAAR5 expressed in HEK293 cells assessed as cAMP accumulation after 20 mins by BRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2019
Entry Details Article
PubMed
TargetTrace amine-associated receptor 5(Mouse)
University of Genoa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50293845BDBM50293845(CHEMBL4169509)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at mouse TAAR5 expressed in HEK293 cells assessed as cAMP accumulation after 20 mins by BRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/5/2020
Entry Details Article
PubMed
TargetTrace amine-associated receptor 5(Mouse)
University of Genoa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50293911BDBM50293911(CHEMBL4177366)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at mouse TAAR5 expressed in HEK293 cells assessed as cAMP accumulation after 20 mins by BRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/5/2020
Entry Details Article
PubMed
TargetTrace amine-associated receptor 5(Mouse)
University of Genoa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50293376BDBM50293376(CHEMBL4163065)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at mouse TAAR5 expressed in HEK293 cells assessed as cAMP accumulation after 20 mins by BRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/5/2020
Entry Details Article
PubMed
TargetTrace amine-associated receptor 5(Mouse)
University of Genoa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50293380BDBM50293380(CHEMBL4173769)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at mouse TAAR5 expressed in HEK293 cells assessed as cAMP accumulation after 20 mins by BRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/5/2020
Entry Details Article
PubMed
TargetTrace amine-associated receptor 5(Mouse)
University of Genoa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50227835BDBM50227835(CHEMBL4096403)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at mouse TAAR5 expressed in HEK293 cells assessed as cAMP accumulation after 20 mins by BRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2019
Entry Details Article
PubMed
TargetTrace amine-associated receptor 5(Mouse)
University of Genoa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50227825BDBM50227825(CHEMBL4060464)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at mouse TAAR5 expressed in HEK293 cells assessed as cAMP accumulation after 20 mins by BRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2019
Entry Details Article
PubMed
TargetTrace amine-associated receptor 5(Mouse)
University of Genoa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50292710BDBM50292710(CHEMBL4161604)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at mouse TAAR5 expressed in HEK293 cells assessed as cAMP accumulation after 20 mins by BRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/5/2020
Entry Details Article
PubMed
TargetTrace amine-associated receptor 5(Mouse)
University of Genoa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50227836BDBM50227836(CHEMBL4076103)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at mouse TAAR5 expressed in HEK293 cells assessed as cAMP accumulation after 20 mins by BRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2019
Entry Details Article
PubMed
TargetTrace amine-associated receptor 5(Mouse)
University of Genoa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50227828BDBM50227828(CHEMBL4068661)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at mouse TAAR5 expressed in HEK293 cells assessed as cAMP accumulation after 20 mins by BRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2019
Entry Details Article
PubMed
TargetTrace amine-associated receptor 5(Mouse)
University of Genoa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50227834BDBM50227834(CHEMBL4077681)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at mouse TAAR5 expressed in HEK293 cells assessed as cAMP accumulation after 20 mins by BRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2019
Entry Details Article
PubMed
TargetTrace amine-associated receptor 5(Mouse)
University of Genoa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50227833BDBM50227833(CHEMBL4088381)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at mouse TAAR5 expressed in HEK293 cells assessed as cAMP accumulation after 20 mins by BRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2019
Entry Details Article
PubMed
TargetTrace amine-associated receptor 5(Mouse)
University of Genoa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50227824BDBM50227824(CHEMBL4088689)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at mouse TAAR5 expressed in HEK293 cells assessed as cAMP accumulation after 20 mins by BRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2019
Entry Details Article
PubMed
TargetTrace amine-associated receptor 5(Mouse)
University of Genoa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50292711BDBM50292711(CHEMBL3628707)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at mouse TAAR5 expressed in HEK293 cells assessed as cAMP accumulation after 20 mins by BRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/5/2020
Entry Details Article
PubMed
TargetTrace amine-associated receptor 5(Mouse)
University of Genoa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50227351BDBM50227351(CHEMBL3628706)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at mouse TAAR5 expressed in HEK293 cells assessed as cAMP accumulation after 20 mins by BRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2019
Entry Details Article
PubMed
TargetTrace amine-associated receptor 5(Mouse)
University of Genoa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50378363BDBM50378363(CHEMBL574656)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at mouse TAAR5 expressed in HEK293 cells assessed as cAMP accumulation after 20 mins by BRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2019
Entry Details Article
PubMed
TargetTrace amine-associated receptor 5(Mouse)
University of Genoa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 18792BDBM18792(Chlorazin | 1-(4-chlorophenyl)-6,6-dimethyl-1,6-di...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at mouse TAAR5 expressed in HEK293 cells assessed as cAMP accumulation after 20 mins by BRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2019
Entry Details Article
PubMed
TargetTrace amine-associated receptor 5(Mouse)
University of Genoa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 18069BDBM18069(CHEMBL22 | TMP | Trimethoprim (TMP) | 5-[(3,4,5-tr...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at mouse TAAR5 expressed in HEK293 cells assessed as cAMP accumulation after 20 mins by BRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2019
Entry Details Article
PubMed
TargetTrace amine-associated receptor 5(Mouse)
University of Genoa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50227839BDBM50227839(CHEMBL4094764)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at mouse TAAR5 expressed in HEK293 cells assessed as cAMP accumulation after 20 mins by BRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2019
Entry Details Article
PubMed
TargetTrace amine-associated receptor 5(Mouse)
University of Genoa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50227838BDBM50227838(CHEMBL4102503)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at mouse TAAR5 expressed in HEK293 cells assessed as cAMP accumulation after 20 mins by BRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2019
Entry Details Article
PubMed
TargetTrace amine-associated receptor 5(Mouse)
University of Genoa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50227841BDBM50227841(ABOB | Moroxydine | SKF-8898A)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at mouse TAAR5 expressed in HEK293 cells assessed as cAMP accumulation after 20 mins by BRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2019
Entry Details Article
PubMed
TargetTrace amine-associated receptor 5(Mouse)
University of Genoa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50227840BDBM50227840(CHEMBL2079013)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at mouse TAAR5 expressed in HEK293 cells assessed as cAMP accumulation after 20 mins by BRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2019
Entry Details Article
PubMed
TargetTrace amine-associated receptor 5(Mouse)
University of Genoa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50293265BDBM50293265(CHEMBL4162640)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at mouse TAAR5 expressed in HEK293 cells assessed as cAMP accumulation after 20 mins by BRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/5/2020
Entry Details Article
PubMed
TargetTrace amine-associated receptor 5(Mouse)
University of Genoa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50293017BDBM50293017(CHEMBL4172905)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at mouse TAAR5 expressed in HEK293 cells assessed as cAMP accumulation after 20 mins by BRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/5/2020
Entry Details Article
PubMed
TargetTrace amine-associated receptor 5(Mouse)
University of Genoa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50293965BDBM50293965(CHEMBL4162232)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at mouse TAAR5 expressed in HEK293 cells assessed as cAMP accumulation after 20 mins by BRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/5/2020
Entry Details Article
PubMed
TargetTrace amine-associated receptor 5(Mouse)
University of Genoa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50053630BDBM50053630(N-(4-methylphenyl)imidodicarbonimidic diamide | 4-...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at mouse TAAR5 expressed in HEK293 cells assessed as cAMP accumulation after 20 mins by BRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2019
Entry Details Article
PubMed
TargetTrace amine-associated receptor 5(Mouse)
University of Genoa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50053596BDBM50053596(1-phenylbiguanide | Phenyl biguanide | N-phenylimi...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at mouse TAAR5 expressed in HEK293 cells assessed as cAMP accumulation after 20 mins by BRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2019
Entry Details Article
PubMed
TargetTrace amine-associated receptor 5(Mouse)
University of Genoa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50053595BDBM50053595(4-Chlorophenylbiguanide | N-(4-chlorophenyl)imidod...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at mouse TAAR5 expressed in HEK293 cells assessed as cAMP accumulation after 20 mins by BRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2019
Entry Details Article
PubMed
TargetTrace amine-associated receptor 5(Mouse)
University of Genoa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50227975BDBM50227975(CHEMBL4087775)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at mouse TAAR5 expressed in HEK293 cells assessed as cAMP accumulation after 20 mins by BRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2019
Entry Details Article
PubMed