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TargetD(1A) dopamine receptor(Mouse)
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Curated by PDSP Ki Database
LigandPNGBDBM82247(SCH 23390,R(+) | CAS_87134-87-0 | CHEMBL2158641 | ...)
Affinity DataKi:  0.140nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2011
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Mouse)
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Curated by PDSP Ki Database
LigandPNGBDBM50026957((cis) 2-{4-[3-(2-Trifluoromethyl-thioxanthen-9-yli...)
Affinity DataKi:  0.320nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2011
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Mouse)
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Curated by PDSP Ki Database
LigandPNGBDBM82247(SCH 23390,R(+) | CAS_87134-87-0 | CHEMBL2158641 | ...)
Affinity DataKi:  0.400nMAssay Description:Binding affinity to displace [3H]- SCH 23390 against Dopamine receptor D1More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Mouse)
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Curated by PDSP Ki Database
LigandPNGBDBM50008735(CHEMBL8514 | BUTACLAMOL,d- | (+)-3-(tert-butyl)-(3...)
Affinity DataKi:  0.950nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2011
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Mouse)
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Curated by PDSP Ki Database
LigandPNGBDBM81986(NSC_173870 | CHEMBL545000 | CAS_173870 | 3-Methyl-...)
Affinity DataKi:  1.90nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2011
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Mouse)
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Curated by PDSP Ki Database
LigandPNGBDBM78433(2-[4-[3-[2-(trifluoromethyl)phenothiazin-10-yl]pro...)
Affinity DataKi:  4.5nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2011
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Mouse)
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Curated by PDSP Ki Database
LigandPNGBDBM22871(13-chloro-10-(4-methylpiperazin-1-yl)-2-oxa-9-azat...)
Affinity DataKi:  16nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2011
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Mouse)
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Curated by PDSP Ki Database
LigandPNGBDBM81985(CAS_42239-60-1 | NSC_172286 | Tilozepine)
Affinity DataKi:  17nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2011
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Mouse)
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Curated by PDSP Ki Database
LigandPNGBDBM50004822(CHEMBL24077 | SKF 38393 (+) | SK-383933 | R(+)SKF ...)
Affinity DataKi:  18nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2011
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Mouse)
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Curated by PDSP Ki Database
LigandPNGBDBM50001888([3-(2-Chloro-phenothiazin-10-yl)-propyl]-dimethyl-...)
Affinity DataKi:  25nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2011
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Mouse)
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Curated by PDSP Ki Database
LigandPNGBDBM22869(6-chloro-10-(4-methylpiperazin-1-yl)-2,9-diazatric...)
Affinity DataKi:  55nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2011
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Mouse)
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Curated by PDSP Ki Database
LigandPNGBDBM50509150(LY-3154207 | Ly3154207 | Mevidalen)
Affinity DataEC50:  62nMAssay Description:Positive allosteric modulator activity at mouse D1 receptor transiently expressed in HEK293 cells assessed as potentiation of EC20 dopamine-induced c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetD(1A) dopamine receptor(Mouse)
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Curated by PDSP Ki Database
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataKi:  76nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2011
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Mouse)
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Curated by PDSP Ki Database
LigandPNGBDBM50040241(CHEMBL63756 | 3-Fluoro-6-(4-methyl-piperazin-1-yl)...)
Affinity DataKi:  85nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2011
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Mouse)
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Curated by PDSP Ki Database
LigandPNGBDBM50001955(APOKYN | CHEMBL53 | (Apomorphine) 6-Methyl-5,6,6a,...)
Affinity DataKi:  101nMAssay Description:Displacement of [3H]SCH23390 from dopamine D1 receptor in mouse Ltk- fibroblast cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Mouse)
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Curated by PDSP Ki Database
LigandPNGBDBM435739(US10611751, Example 1 | 2-(2,6-dichlorophenyl)-1-(...)
Affinity DataEC50:  151nMAssay Description:Positive allosteric modulation of mouse D1 receptor expressed in HEK293 cells assessed as increase in cyclic AMP production measured after 60 mins in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetD(1A) dopamine receptor(Mouse)
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Curated by PDSP Ki Database
LigandPNGBDBM21342((4R,7R)-N,N-diethyl-6-methyl-6,11-diazatetracyclo[...)
Affinity DataKi:  180nMAssay Description:Binding affinities towards Dopamine receptor D1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetD(1A) dopamine receptor(Mouse)
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Curated by PDSP Ki Database
LigandPNGBDBM50118576((2,4-Dimethyl-azetidin-1-yl)-(7-methyl-4,6,6a,7,8,...)
Affinity DataKi:  230nMAssay Description:Binding affinity against Dopamine receptor D1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Mouse)
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Curated by PDSP Ki Database
LigandPNGBDBM50118579((2,4-Dimethyl-azetidin-1-yl)-(7-methyl-4,6,6a,7,8,...)
Affinity DataKi:  290nMAssay Description:Binding affinity towards Dopamine receptor D1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Mouse)
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Curated by PDSP Ki Database
LigandPNGBDBM50509151(CHEMBL3421730)
Affinity DataEC50:  312nMAssay Description:Positive allosteric modulation of mouse D1R expressed in HEK293 cells assessed as increase in dopamine-induced cAMP accumulation after 60 mins by HTR...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Mouse)
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Curated by PDSP Ki Database
LigandPNGBDBM50118577((2,4-Dimethyl-azetidin-1-yl)-(7-methyl-4,6,6a,7,8,...)
Affinity DataKi:  340nMAssay Description:Binding affinity towards Dopamine receptor D1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Mouse)
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Curated by PDSP Ki Database
LigandPNGBDBM21397(8-[4-(4-fluorophenyl)-4-oxidanylidene-butyl]-1-phe...)
Affinity DataKi:  360nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2011
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Mouse)
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Curated by PDSP Ki Database
LigandPNGBDBM50028421(Permax | CHEMBL1275 | Pergolide | 9-Methylsulfanyl...)
Affinity DataKi:  400nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2011
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Mouse)
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Curated by PDSP Ki Database
LigandPNGBDBM50026957((cis) 2-{4-[3-(2-Trifluoromethyl-thioxanthen-9-yli...)
Affinity DataKi:  474nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2011
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Mouse)
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Curated by PDSP Ki Database
LigandPNGBDBM81777(NPA,(+) | NPA | CAS_132-66-1 | NSC_8594 | NPA,(-))
Affinity DataKi:  480nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2011
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Mouse)
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Curated by PDSP Ki Database
LigandPNGBDBM50060965(2-[2-((3aR,9bR)-6-Methoxy-1,3,3a,4,5,9b-hexahydro-...)
Affinity DataKi:  717nMAssay Description:Binding affinity against Dopamine receptor D1 using [3H]SCH-23390 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Mouse)
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Curated by PDSP Ki Database
LigandPNGBDBM50034043(CHEMBL14376 | 1-(4-{3-[4-(6-Fluoro-benzo[d]isoxazo...)
Affinity DataIC50: 750nMAssay Description:Binding affinity against Dopamine receptor D1 was determined using [3H]SCH-23390 radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/31/2012
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Mouse)
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Curated by PDSP Ki Database
LigandPNGBDBM50132693(4-Amino-N-(1-benzyl-piperidin-4-yl)-5-chloro-2-met...)
Affinity DataKi:  820nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2011
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Mouse)
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Curated by PDSP Ki Database
LigandPNGBDBM50001859(BUSPAR | CHEMBL49 | 8-[4-(4-Pyrimidin-2-yl-piperaz...)
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity against Dopamine receptor D1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Mouse)
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Curated by PDSP Ki Database
LigandPNGBDBM50007674((+)-erythro 4-[2-(4-Benzyl-piperidin-1-yl)-1-hydro...)
Affinity DataIC50: 1.00E+3nMAssay Description:Compound was tested for the binding affinity against dopamine receptor D1 by using [3H]-SCH- 23390 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Mouse)
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Curated by PDSP Ki Database
LigandPNGBDBM50002218(CHEMBL42228 | CHEMBL543412 | 2-(1-Cyclopropylmethy...)
Affinity DataKi: >1.00E+3nMAssay Description:The compound was tested in vitro for its binding affinity towards dopamine receptor D1More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Mouse)
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Curated by PDSP Ki Database
LigandPNGBDBM50014154(CHEMBL38465 | 2-(5-Methyl-1H-imidazol-4-ylmethyl)-...)
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity for Dopamine receptor D1 was determined by using [3H]SCH-23390 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2012
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Mouse)
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Curated by PDSP Ki Database
LigandPNGBDBM21393(cid_1220 | CHEMBL56 | 7-(dipropylamino)-5,6,7,8-te...)
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity against Dopamine receptor D1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Mouse)
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Curated by PDSP Ki Database
LigandPNGBDBM186927(US9079895, 19s)
Affinity DataKi:  1.35E+3nMpH: 7.4Assay Description:The detailed experimental protocols for the radioligand and functional receptor assays are available on the NIMH PDSP website at http://pdsp.med.unc....More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2016
Entry Details
US Patent

TargetD(1A) dopamine receptor(Mouse)
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Curated by PDSP Ki Database
LigandPNGBDBM186935(US9079895, 23s)
Affinity DataKi:  2.04E+3nMpH: 7.4Assay Description:The detailed experimental protocols for the radioligand and functional receptor assays are available on the NIMH PDSP website at http://pdsp.med.unc....More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2016
Entry Details
US Patent

TargetD(1A) dopamine receptor(Mouse)
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Curated by PDSP Ki Database
LigandPNGBDBM50251327((R)-2-Butoxy-6-methyl-5,6,6a,7-tetrahydro-4H-diben...)
Affinity DataKi:  2.10E+3nMAssay Description:Displacement of [3H]SCH23390 from dopamine D1 receptor in mouse Ltk- fibroblast cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Mouse)
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Curated by PDSP Ki Database
LigandPNGBDBM86525(NSC_77445 | CHEMBL79834 | CAS_77445 | AMI-193)
Affinity DataKi:  2.53E+3nMAssay Description:Tested for binding affinity against dopamine receptor D1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Mouse)
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Curated by PDSP Ki Database
LigandPNGBDBM50251320((R)-2-Ethoxy-6-methyl-5,6,6a,7-tetrahydro-4H-diben...)
Affinity DataKi:  2.90E+3nMAssay Description:Displacement of [3H]SCH23390 from dopamine D1 receptor in mouse Ltk- fibroblast cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Mouse)
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Curated by PDSP Ki Database
LigandPNGBDBM50251321((R)-6-Methyl-2-propoxy-5,6,6a,7-tetrahydro-4H-dibe...)
Affinity DataKi:  3.50E+3nMAssay Description:Displacement of [3H]SCH23390 from dopamine D1 receptor in mouse Ltk- fibroblast cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Mouse)
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Curated by PDSP Ki Database
LigandPNGBDBM81873(NSC_55397 | CAS_55397 | QUINPIROLE | LY-171555)
Affinity DataKi:  5.00E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2011
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Mouse)
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Curated by PDSP Ki Database
LigandPNGBDBM50251330(1,2-Bis-[R-(-)-apomorphine-2'-oxy]ethane | CHEMBL4...)
Affinity DataKi:  5.20E+3nMAssay Description:Displacement of [3H]SCH23390 from dopamine D1 receptor in mouse Ltk- fibroblast cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Mouse)
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Curated by PDSP Ki Database
LigandPNGBDBM50251328([R-(-)-Apomorphine-2-yl]-(2'-hydroxy-ethyl)ether |...)
Affinity DataKi:  5.30E+3nMAssay Description:Displacement of [3H]SCH23390 from dopamine D1 receptor in mouse Ltk- fibroblast cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Mouse)
Novo Industri

Curated by PDSP Ki Database
LigandPNGBDBM186942(US9079895, 27s)
Affinity DataKi:  5.85E+3nMpH: 7.4Assay Description:The detailed experimental protocols for the radioligand and functional receptor assays are available on the NIMH PDSP website at http://pdsp.med.unc....More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2016
Entry Details
US Patent

TargetD(1A) dopamine receptor(Mouse)
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Curated by PDSP Ki Database
LigandPNGBDBM50251329(2-{[R-(-)-Apomorphine-2'-oxy]ethoxy}-ethanol | CHE...)
Affinity DataKi:  7.60E+3nMAssay Description:Displacement of [3H]SCH23390 from dopamine D1 receptor in mouse Ltk- fibroblast cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Mouse)
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Curated by PDSP Ki Database
LigandPNGBDBM186937(US9079895, 25s)
Affinity DataKi:  8.37E+3nMpH: 7.4Assay Description:The detailed experimental protocols for the radioligand and functional receptor assays are available on the NIMH PDSP website at http://pdsp.med.unc....More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2016
Entry Details
US Patent

TargetD(1A) dopamine receptor(Mouse)
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Curated by PDSP Ki Database
LigandPNGBDBM186953(US9079895, 60)
Affinity DataKi: >1.00E+4nMpH: 7.4Assay Description:The detailed experimental protocols for the radioligand and functional receptor assays are available on the NIMH PDSP website at http://pdsp.med.unc....More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2016
Entry Details
US Patent

TargetD(1A) dopamine receptor(Mouse)
Novo Industri

Curated by PDSP Ki Database
LigandPNGBDBM50002245(CHEMBL130356 | CHEMBL137776 | 4-[2-(1-Cyclopropylm...)
Affinity DataKi: >1.00E+4nMAssay Description:The compound was tested in vitro for its binding affinity towards dopamine receptor D1More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/23/2012
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Mouse)
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Curated by PDSP Ki Database
LigandPNGBDBM50108659(1'-benzyl-3-methoxyspiro[1,3-dihydroisobenzofuran-...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of SCH 23390 binding to Dopamine receptor D1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Mouse)
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Curated by PDSP Ki Database
LigandPNGBDBM50251331(Bis-{[R-(-)-apomorphine-2-oxy]ethyl} ether | CHEMB...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]SCH23390 from dopamine D1 receptor in mouse Ltk- fibroblast cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Mouse)
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Curated by PDSP Ki Database
LigandPNGBDBM186968(US9079895, 70)
Affinity DataKi: >1.00E+4nMpH: 7.4Assay Description:The detailed experimental protocols for the radioligand and functional receptor assays are available on the NIMH PDSP website at http://pdsp.med.unc....More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2016
Entry Details
US Patent

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