Compile Data Set for Download or QSAR
Report error Found 725 of affinity data for UniProtKB/TrEMBL: Q63931
TargetCholecystokinin receptor type A(Guinea pig)
Hadassah-University Hospital

Curated by ChEMBL
LigandPNGBDBM50004436(3-Acetylamino-N-[1-[1-({[1-{1-[1-(1-carbamoyl-2-ph...)
Affinity DataEC50:  0.100nMAssay Description:In vitro smooth muscle contraction activity in guinea pig gall bladder cholecystokinin type A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Guinea pig)
Hadassah-University Hospital

Curated by ChEMBL
LigandPNGBDBM50016504(Boc-Tyr(SO3Na)-gNle-mGIy-Trp-(N-Me)Nle-Asp-Phe-NH2...)
Affinity DataKi:  0.230nMAssay Description:The compound was tested for the inhibition of [3H]propionyl specific binding to Cholecystokinin 8 receptor of guinea pig brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Guinea pig)
Hadassah-University Hospital

Curated by ChEMBL
LigandPNGBDBM21147((3S)-3-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-[(3S)-3-...)
Affinity DataKi:  0.280nMAssay Description:Inhibition of [3H]pCCK-8 binding to Cholecystokinin type A receptor of Guinea pig pancreatic membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Guinea pig)
Hadassah-University Hospital

Curated by ChEMBL
LigandPNGBDBM21147((3S)-3-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-[(3S)-3-...)
Affinity DataKi:  0.280nMAssay Description:Displacement of 0.1 nM [3H]Boc[Nle28,31]-CCK27-33 from guinea pig pancreatic membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Guinea pig)
Hadassah-University Hospital

Curated by ChEMBL
LigandPNGBDBM21147((3S)-3-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-[(3S)-3-...)
Affinity DataKi:  0.280nMAssay Description:The compound was tested for the inhibition of [3H]propionyl specific binding to CCK-8 receptor of guinea pig brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Guinea pig)
Hadassah-University Hospital

Curated by ChEMBL
LigandPNGBDBM21147((3S)-3-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-[(3S)-3-...)
Affinity DataIC50: 0.280nMAssay Description:Displacement of [125I]Bolton-Hunter-CCK-8 from guinea pig pancreas Cholecystokinin type A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetCholecystokinin receptor type A(Guinea pig)
Hadassah-University Hospital

Curated by ChEMBL
LigandPNGBDBM50016504(Boc-Tyr(SO3Na)-gNle-mGIy-Trp-(N-Me)Nle-Asp-Phe-NH2...)
Affinity DataKi:  0.310nMAssay Description:Ability to displace 1 nM [3H]pCCK-8 from Cholecystokinin type A receptor in guinea pig pancreatic membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2012
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Guinea pig)
Hadassah-University Hospital

Curated by ChEMBL
LigandPNGBDBM21147((3S)-3-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-[(3S)-3-...)
Affinity DataIC50: 0.400nMAssay Description:Displacement of [125I]BH-CCK-8 from Cholecystokinin type A receptor in guinea pig pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2012
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Guinea pig)
Hadassah-University Hospital

Curated by ChEMBL
LigandPNGBDBM50004477(N-(1-Carbamoyl-2-phenyl-ethyl)-3-({2-[3-(1H-indol-...)
Affinity DataIC50: 0.5nMAssay Description:In vitro ability to inhibit [125I]Bolton-Hunter-CCK-8 binding to Cholecystokinin type A receptor in guinea pig pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Guinea pig)
Hadassah-University Hospital

Curated by ChEMBL
LigandPNGBDBM21147((3S)-3-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-[(3S)-3-...)
Affinity DataKi:  0.600nMAssay Description:Ability to displace 1 nM [3H]pCCK-8 from Cholecystokinin type A receptor in guinea pig pancreatic membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2012
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Guinea pig)
Hadassah-University Hospital

Curated by ChEMBL
LigandPNGBDBM21147((3S)-3-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-[(3S)-3-...)
Affinity DataKi:  0.640nMAssay Description:Tested for the inhibition of [3H]pCCK-8 binding to Cholecystokinin type A receptor in pancreatic membranes of guinea-pigMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetCholecystokinin receptor type A(Guinea pig)
Hadassah-University Hospital

Curated by ChEMBL
LigandPNGBDBM21147((3S)-3-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-[(3S)-3-...)
Affinity DataKi:  0.640nMAssay Description:The compound was tested for the inhibition of [3H]propionyl specific binding to CCK-8 receptor of guinea pig pancreatic membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Guinea pig)
Hadassah-University Hospital

Curated by ChEMBL
LigandPNGBDBM50004480(CHEMBL316944 | CCK7 analogue)
Affinity DataIC50: 0.670nMAssay Description:Evaluated in vitro for its binding affinity towards cholecystokinin type A receptor of guinea pig pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Guinea pig)
Hadassah-University Hospital

Curated by ChEMBL
LigandPNGBDBM21147((3S)-3-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-[(3S)-3-...)
Affinity DataKi:  0.700nMAssay Description:Compound was tested for binding affinity against CCK1 (cholecystokinin) receptor on guinea pig pancreatic membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Guinea pig)
Hadassah-University Hospital

Curated by ChEMBL
LigandPNGBDBM50092398((S)-3-((S)-2-{[(S)-2-tert-Butoxycarbonylamino-3-(1...)
Affinity DataKi: >0.700nMAssay Description:Affinity against Cholecystokinin type A receptor on guinea pig pancreatic membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Guinea pig)
Hadassah-University Hospital

Curated by ChEMBL
LigandPNGBDBM21147((3S)-3-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-[(3S)-3-...)
Affinity DataKi:  0.700nMAssay Description:Affinity of compound on binding of [3H]pCCK-8 to the cholecystokinin type A receptor in guinea pig pancreatic membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2012
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Guinea pig)
Hadassah-University Hospital

Curated by ChEMBL
LigandPNGBDBM50092405((S)-N-((S)-1-Carbamoyl-2-phenyl-ethyl)-3-((S)-2-{[...)
Affinity DataKi: >0.700nMAssay Description:Affinity against Cholecystokinin type A receptor on guinea pig pancreatic membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Guinea pig)
Hadassah-University Hospital

Curated by ChEMBL
LigandPNGBDBM50092405((S)-N-((S)-1-Carbamoyl-2-phenyl-ethyl)-3-((S)-2-{[...)
Affinity DataKi:  0.75nMAssay Description:Ability to displace 1 nM [3H]pCCK-8 from Cholecystokinin type A receptor in guinea pig pancreatic membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2012
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Guinea pig)
Hadassah-University Hospital

Curated by ChEMBL
LigandPNGBDBM50004474(CHEMBL316949 | N-(1-Carbamoyl-2-phenyl-ethyl)-3-{2...)
Affinity DataIC50: 0.770nMAssay Description:Evaluated in vitro for its binding affinity towards cholecystokinin type A receptor of guinea pig pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Guinea pig)
Hadassah-University Hospital

Curated by ChEMBL
LigandPNGBDBM50004474(CHEMBL316949 | N-(1-Carbamoyl-2-phenyl-ethyl)-3-{2...)
Affinity DataIC50: 0.770nMAssay Description:In vitro ability to inhibit [125I]Bolton-Hunter-CCK-8 binding to Cholecystokinin type A receptor in guinea pig pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Guinea pig)
Hadassah-University Hospital

Curated by ChEMBL
LigandPNGBDBM50016504(Boc-Tyr(SO3Na)-gNle-mGIy-Trp-(N-Me)Nle-Asp-Phe-NH2...)
Affinity DataKi:  0.930nMAssay Description:The compound was tested for the inhibition of [3H]propionyl specific binding to Cholecystokinin 8 receptor of guinea pig pancreatic membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Guinea pig)
Hadassah-University Hospital

Curated by ChEMBL
LigandPNGBDBM50016425(3-{2-[2-(2-{2-[2-(tert-Butoxycarbonyl-methyl-amino...)
Affinity DataKi:  0.930nMAssay Description:Displacement of 0.1 nM [3H]Boc[Nle28,31]-CCK27-33 from guinea pig pancreatic membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Guinea pig)
Hadassah-University Hospital

Curated by ChEMBL
LigandPNGBDBM50016425(3-{2-[2-(2-{2-[2-(tert-Butoxycarbonyl-methyl-amino...)
Affinity DataIC50: 0.930nMAssay Description:In vitro ability to inhibit [3H]propionyl-CCK-8 binding to Cholecystokinin type A receptor in guinea pig pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Guinea pig)
Hadassah-University Hospital

Curated by ChEMBL
LigandPNGBDBM50004482(CCK7 analogue | CHEMBL263742 | N-(1-Carbamoyl-2-ph...)
Affinity DataIC50: 0.990nMAssay Description:In vitro ability to inhibit [125I]Bolton-Hunter-CCK-8 binding to Cholecystokinin type A receptor in guinea pig pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Guinea pig)
Hadassah-University Hospital

Curated by ChEMBL
LigandPNGBDBM50283831(N-tert-Butyl-2-[(3R,5S,7R)-7-(3-fluoro-phenyl)-2-o...)
Affinity DataIC50: 1nMAssay Description:Inhibitory activity against cholecystokinin-A (CCK-A) receptor in pancreas of guinea pig.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetCholecystokinin receptor type A(Guinea pig)
Hadassah-University Hospital

Curated by ChEMBL
LigandPNGBDBM50283843(N-(2-Chloro-phenyl)-2-[(3R,5S,7R)-2-oxo-7-phenyl-5...)
Affinity DataIC50: 1.10nMAssay Description:Inhibitory activity against cholecystokinin-A (CCK-A) receptor in pancreas of guinea pig.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetCholecystokinin receptor type A(Guinea pig)
Hadassah-University Hospital

Curated by ChEMBL
LigandPNGBDBM50283832(N-tert-Butyl-2-[(3R,5S,7R)-2-oxo-7-phenyl-5-p-toly...)
Affinity DataIC50: 1.10nMAssay Description:Inhibitory activity against cholecystokinin-A (CCK-A) receptor in pancreas of guinea pig.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetCholecystokinin receptor type A(Guinea pig)
Hadassah-University Hospital

Curated by ChEMBL
LigandPNGBDBM50044039((S)-N-((S)-1-Carbamoyl-2-phenyl-ethyl)-3-[(S)-2-[(...)
Affinity DataIC50: 1.10nMAssay Description:Inhibition of [125I]Bolton-Hunter CCK-8 binding to cholecystokinin type A receptor in guinea pig pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Guinea pig)
Hadassah-University Hospital

Curated by ChEMBL
LigandPNGBDBM50283845(2-[(3R,5S,7R)-2-Oxo-7-phenyl-5-o-tolyl-3-(3-m-toly...)
Affinity DataIC50: 1.10nMAssay Description:Inhibitory activity against cholecystokinin-A (CCK-A) receptor in pancreas of guinea pig.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetCholecystokinin receptor type A(Guinea pig)
Hadassah-University Hospital

Curated by ChEMBL
LigandPNGBDBM50004440(3-Acetylamino-N-[1-[1-({[1-{1-[1-(1-carbamoyl-2-ph...)
Affinity DataEC50:  1.20nMAssay Description:In vitro smooth muscle contraction activity in guinea pig gall bladder cholecystokinin type A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Guinea pig)
Hadassah-University Hospital

Curated by ChEMBL
LigandPNGBDBM50044033((S)-3-[(S)-2-((S)-2-Benzoylamino-3-1H-indol-3-yl-p...)
Affinity DataIC50: 1.30nMAssay Description:Inhibition of [125I]Bolton-Hunter CCK-8 binding to cholecystokinin type A receptor in guinea pig pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Guinea pig)
Hadassah-University Hospital

Curated by ChEMBL
LigandPNGBDBM50283842(N-tert-Butyl-2-[(3R,5S,7R)-2-oxo-7-phenyl-5-m-toly...)
Affinity DataIC50: 1.30nMAssay Description:Inhibitory activity against cholecystokinin-A (CCK-A) receptor in pancreas of guinea pig.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetCholecystokinin receptor type A(Guinea pig)
Hadassah-University Hospital

Curated by ChEMBL
LigandPNGBDBM50092388(3-(2-{[2-(3-tert-Butoxycarbonylamino-propionylamin...)
Affinity DataKi:  1.35nMAssay Description:Affinity against Cholecystokinin type A receptor on guinea pig pancreatic membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Guinea pig)
Hadassah-University Hospital

Curated by ChEMBL
LigandPNGBDBM50004439(3-Acetylamino-N-[1-[1-({[1-{1-[1-(1-carbamoyl-2-ph...)
Affinity DataEC50:  1.40nMAssay Description:In vitro smooth muscle contraction activity in guinea pig gall bladder cholecystokinin type A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Guinea pig)
Hadassah-University Hospital

Curated by ChEMBL
LigandPNGBDBM50044042((S)-N-((S)-1-Carbamoyl-2-phenyl-ethyl)-3-[(S)-2-[2...)
Affinity DataIC50: 1.40nMAssay Description:Inhibition of [125I]Bolton-Hunter CCK-8 binding to cholecystokinin type A receptor in guinea pig pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Guinea pig)
Hadassah-University Hospital

Curated by ChEMBL
LigandPNGBDBM50044028((S)-N-((S)-1-Carbamoyl-2-phenyl-ethyl)-3-[(S)-2-((...)
Affinity DataIC50: 1.60nMAssay Description:Inhibition of [125I]Bolton-Hunter CCK-8 binding to cholecystokinin type A receptor in guinea pig pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Guinea pig)
Hadassah-University Hospital

Curated by ChEMBL
LigandPNGBDBM50283838(N-tert-Butyl-2-[(3R,5S,7R)-2-oxo-5-phenyl-7-m-toly...)
Affinity DataIC50: 1.60nMAssay Description:Inhibitory activity against cholecystokinin-A (CCK-A) receptor in pancreas of guinea pig.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetCholecystokinin receptor type A(Guinea pig)
Hadassah-University Hospital

Curated by ChEMBL
LigandPNGBDBM50044038((S)-N-((S)-1-Carbamoyl-2-phenyl-ethyl)-3-[(S)-2-[(...)
Affinity DataIC50: 1.70nMAssay Description:Inhibition of [125I]Bolton-Hunter CCK-8 binding to cholecystokinin type A receptor in guinea pig pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Guinea pig)
Hadassah-University Hospital

Curated by ChEMBL
LigandPNGBDBM50016506(Sodium; (4-{2-(2-acetylamino-3-carboxy-propionylam...)
Affinity DataKi:  1.70nMAssay Description:The compound was tested for the inhibition of [3H]propionyl specific binding to Cholecystokinin 8 receptor of guinea pig pancreatic membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Guinea pig)
Hadassah-University Hospital

Curated by ChEMBL
LigandPNGBDBM50283826(N-tert-Butyl-2-{(3R,5S,7R)-3-[3-(3-fluoro-phenyl)-...)
Affinity DataIC50: 1.80nMAssay Description:Inhibitory activity against cholecystokinin-A (CCK-A) receptor in pancreas of guinea pig.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetCholecystokinin receptor type A(Guinea pig)
Hadassah-University Hospital

Curated by ChEMBL
LigandPNGBDBM50044044((S)-N-((S)-1-Carbamoyl-2-phenyl-ethyl)-3-[(S)-2-((...)
Affinity DataIC50: 2nMAssay Description:Inhibition of [125I]Bolton-Hunter CCK-8 binding to cholecystokinin type A receptor in guinea pig pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Guinea pig)
Hadassah-University Hospital

Curated by ChEMBL
LigandPNGBDBM81962(S-L-365,260)
Affinity DataIC50: 2nMAssay Description:Inhibition of binding of [125I]- CCK-33 to guinea pig cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Guinea pig)
Hadassah-University Hospital

Curated by ChEMBL
LigandPNGBDBM50004437(3-Acetylamino-N-[1-[1-({[1-(1-{[1-(1-carbamoyl-2-p...)
Affinity DataEC50:  2nMAssay Description:In vitro smooth muscle contraction activity in guinea pig gall bladder cholecystokinin type A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Guinea pig)
Hadassah-University Hospital

Curated by ChEMBL
LigandPNGBDBM50092391(3-(2-{[2-(2-Carbamoyl-acetylamino)-3-(1H-indol-3-y...)
Affinity DataKi:  2.05nMAssay Description:Affinity against Cholecystokinin type A receptor on guinea pig pancreatic membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Guinea pig)
Hadassah-University Hospital

Curated by ChEMBL
LigandPNGBDBM50421963(CHEMBL2310856)
Affinity DataIC50: 2.10nMAssay Description:Evaluated in vitro for its binding affinity towards cholecystokinin type A receptor of guinea pig pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Guinea pig)
Hadassah-University Hospital

Curated by ChEMBL
LigandPNGBDBM50044032((S)-N-((S)-1-Carbamoyl-2-phenyl-ethyl)-3-[(S)-2-[(...)
Affinity DataIC50: 2.20nMAssay Description:Inhibition of [125I]Bolton-Hunter CCK-8 binding to cholecystokinin type A receptor in guinea pig pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Guinea pig)
Hadassah-University Hospital

Curated by ChEMBL
LigandPNGBDBM50283827(N-tert-Butyl-2-{(3R,5S,7R)-3-[3-(4-methoxy-phenyl)...)
Affinity DataIC50: 2.20nMAssay Description:Inhibitory activity against cholecystokinin-A (CCK-A) receptor in pancreas of guinea pig.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetCholecystokinin receptor type A(Guinea pig)
Hadassah-University Hospital

Curated by ChEMBL
LigandPNGBDBM50044037((S)-N-((S)-1-Carbamoyl-2-phenyl-ethyl)-3-[(S)-2-((...)
Affinity DataIC50: 2.30nMAssay Description:Inhibition of [125I]Bolton-Hunter CCK-8 binding to cholecystokinin type A receptor in guinea pig pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Guinea pig)
Hadassah-University Hospital

Curated by ChEMBL
LigandPNGBDBM50092396(3-(2-{[2-Amino-3-(1H-indol-3-yl)-propionyl]-methyl...)
Affinity DataKi:  2.60nMAssay Description:Affinity against Cholecystokinin type A receptor on guinea pig pancreatic membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Guinea pig)
Hadassah-University Hospital

Curated by ChEMBL
LigandPNGBDBM50092398((S)-3-((S)-2-{[(S)-2-tert-Butoxycarbonylamino-3-(1...)
Affinity DataKi:  2.60nMAssay Description:Ability to displace 1 nM [3H]pCCK-8 from Cholecystokinin type A receptor in guinea pig pancreatic membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2012
Entry Details Article
PubMed
Displayed 1 to 50 (of 725 total ) | Next | Last >>
Jump to: