Compile Data Set for Download or QSAR
Report error Found 231 of affinity data for UniProtKB/TrEMBL: Q7Z601
TargetProbable G-protein coupled receptor 142(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50437420(CHEMBL2409014)
Affinity DataEC50:  0.200nMAssay Description:Agonist activity at human GPR142 transfected in HEK293 cells after 1 hr by inositol phosphate accumulation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 142(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50437419(CHEMBL2409009)
Affinity DataEC50:  1nMAssay Description:Agonist activity at human GPR142 transfected in HEK293 cells after 1 hr by inositol phosphate accumulation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 142(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50437418(CHEMBL2409011)
Affinity DataEC50:  1nMAssay Description:Agonist activity at human GPR142 transfected in HEK293 cells after 1 hr by inositol phosphate accumulation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 142(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50437417(CHEMBL2409019)
Affinity DataEC50:  1.30nMAssay Description:Agonist activity at human GPR142 transfected in HEK293 cells after 1 hr by inositol phosphate accumulation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 142(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50437416(CHEMBL2409031)
Affinity DataEC50:  5nMAssay Description:Agonist activity at human GPR142 transfected in HEK293 cells after 1 hr by inositol phosphate accumulation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 142(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50437415(CHEMBL2409027)
Affinity DataEC50:  7nMAssay Description:Agonist activity at human GPR142 transfected in HEK293 cells after 1 hr by inositol phosphate accumulation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 142(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50544800(CHEMBL4647745)
Affinity DataEC50:  11nMAssay Description:Agonist activity at human GPR142 receptor expressed in HEK293 cells assessed as accumulation of inositol phosphate incubated for 1 hr followed by IP1...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 142(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50201607(CHEMBL3905835)
Affinity DataEC50:  12nMAssay Description:Agonist activity at human GPR142 expressed in CHO cells measured after 30 to 60 mins by IP-One assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/1/2018
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 142(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50544801(CHEMBL4647456)
Affinity DataEC50:  14nMAssay Description:Agonist activity at human GPR142 receptor expressed in HEK293 cells assessed as accumulation of inositol phosphate incubated for 1 hr followed by IP1...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 142(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50201577(CHEMBL3967871)
Affinity DataEC50:  14nMAssay Description:Agonist activity at human GPR142 expressed in CHO cells measured after 30 to 60 mins by IP-One assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/1/2018
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 142(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50437414(CHEMBL2409023)
Affinity DataEC50:  14nMAssay Description:Agonist activity at human GPR142 transfected in HEK293 cells after 1 hr by inositol phosphate accumulation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 142(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50544805(CHEMBL4646017)
Affinity DataEC50:  14nMAssay Description:Agonist activity at human GPR142 receptor expressed in HEK293 cells assessed as accumulation of inositol phosphate incubated for 1 hr followed by IP1...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 142(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50201604(CHEMBL3976574)
Affinity DataEC50:  16nMAssay Description:Agonist activity at human GPR142 expressed in CHO cells measured after 30 to 60 mins by IP-One assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/1/2018
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 142(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50544804(CHEMBL4637374)
Affinity DataEC50:  16nMAssay Description:Agonist activity at human GPR142 receptor expressed in HEK293 cells assessed as accumulation of inositol phosphate incubated for 1 hr followed by IP1...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 142(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50437413(CHEMBL2409007)
Affinity DataEC50:  22nMAssay Description:Agonist activity at human GPR142 transfected in HEK293 cells after 1 hr by inositol phosphate accumulation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 142(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50201572(CHEMBL3965469)
Affinity DataEC50:  24nMAssay Description:Agonist activity at human GPR142 expressed in CHO cells measured for 3 to 5 mins by Fluo-4AM dye-based FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/1/2018
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 142(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50201572(CHEMBL3965469)
Affinity DataEC50:  24nMAssay Description:Agonist activity at human GPR142 expressed in CHO cells measured after 30 to 60 mins by IP-One assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/1/2018
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 142(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50201607(CHEMBL3905835)
Affinity DataEC50:  25nMAssay Description:Agonist activity at human GPR142 expressed in CHO cells measured for 3 to 5 mins by Fluo-4AM dye-based FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/1/2018
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 142(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50437412(CHEMBL2409021)
Affinity DataEC50:  25nMAssay Description:Agonist activity at human GPR142 transfected in HEK293 cells after 1 hr by inositol phosphate accumulation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 142(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50201604(CHEMBL3976574)
Affinity DataEC50:  26nMAssay Description:Agonist activity at human GPR142 expressed in CHO cells measured for 3 to 5 mins by Fluo-4AM dye-based FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/1/2018
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 142(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50440696(CHEMBL2430979)
Affinity DataEC50:  26nMAssay Description:Agonist activity at human GPR142 expressed in HEK293 cells assessed as inositol phosphate accumulation using [3H]-inositol after 1 hr by scintillatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 142(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM332764(US10196385, Example 3 | Cis-(chiral)-3-Chloro-N-[2...)
Affinity DataEC50:  27nMAssay Description:Agonist activity at human GPR142 receptor expressed in HEK293 cells assessed as accumulation of inositol phosphate incubated for 1 hr followed by IP1...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 142(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM332764(US10196385, Example 3 | Cis-(chiral)-3-Chloro-N-[2...)
Affinity DataEC50:  27.2nMAssay Description:HEK293 cells expressing human GPR142 are maintained in DMEM supplemented with 10% FBS and 800 μg/ml G418 (Geneticin) at 37° C. and 5% CO2. The c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2019
Entry Details
US Patent

TargetProbable G-protein coupled receptor 142(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50437411(CHEMBL2409022)
Affinity DataEC50:  28nMAssay Description:Agonist activity at human GPR142 transfected in HEK293 cells after 1 hr by inositol phosphate accumulation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 142(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50437410(CHEMBL2409030)
Affinity DataEC50:  30nMAssay Description:Agonist activity at human GPR142 transfected in HEK293 cells after 1 hr by inositol phosphate accumulation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 142(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50437409(CHEMBL2409012)
Affinity DataEC50:  30nMAssay Description:Agonist activity at human GPR142 transfected in HEK293 cells after 1 hr by inositol phosphate accumulation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 142(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50544789(CHEMBL4647315)
Affinity DataEC50:  30nMAssay Description:Agonist activity at human GPR142 receptor expressed in HEK293 cells assessed as accumulation of inositol phosphate incubated for 1 hr followed by IP1...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 142(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM332763(US10196385, Example 2 | Cis-(chiral)-N-[2-[5-(1,4-...)
Affinity DataEC50:  30nMAssay Description:Agonist activity at human GPR142 receptor expressed in HEK293 cells assessed as accumulation of inositol phosphate incubated for 1 hr followed by IP1...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 142(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM332763(US10196385, Example 2 | Cis-(chiral)-N-[2-[5-(1,4-...)
Affinity DataEC50:  30.1nMAssay Description:HEK293 cells expressing human GPR142 are maintained in DMEM supplemented with 10% FBS and 800 μg/ml G418 (Geneticin) at 37° C. and 5% CO2. The c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2019
Entry Details
US Patent

TargetProbable G-protein coupled receptor 142(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50201575(CHEMBL3903475)
Affinity DataEC50:  32nMAssay Description:Agonist activity at human GPR142 expressed in CHO cells measured after 30 to 60 mins by IP-One assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/1/2018
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 142(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50544807(CHEMBL4641575)
Affinity DataEC50:  32nMAssay Description:Agonist activity at human GPR142 receptor expressed in HEK293 cells assessed as accumulation of inositol phosphate incubated for 1 hr followed by IP1...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 142(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50201577(CHEMBL3967871)
Affinity DataEC50:  34nMAssay Description:Agonist activity at human GPR142 expressed in CHO cells measured for 3 to 5 mins by Fluo-4AM dye-based FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/1/2018
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 142(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50544810(CHEMBL4641984)
Affinity DataEC50:  35nMAssay Description:Agonist activity at human GPR142 receptor expressed in HEK293 cells assessed as accumulation of inositol phosphate incubated for 1 hr followed by IP1...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 142(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50395775(CHEMBL2164857)
Affinity DataEC50:  36nMAssay Description:Agonist activity at human GPR142 expressed in HEK293 cells assessed as inositol phosphate accumulation after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 142(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50440713(CHEMBL2430977)
Affinity DataEC50:  37nMAssay Description:Agonist activity at human GPR142 expressed in HEK293 cells assessed as inositol phosphate accumulation using [3H]-inositol after 1 hr by scintillatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 142(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50558172(CHEMBL4750179)
Affinity DataIC50: 37nMAssay Description:Agonist activity at human GPR142 expressed in CHO cells measured for 3 mins by Fluo-4M dye based FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 142(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50440714(CHEMBL2431062)
Affinity DataEC50:  37nMAssay Description:Agonist activity at human GPR142 expressed in HEK293 cells assessed as inositol phosphate accumulation using [3H]-inositol after 1 hr by scintillatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 142(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50201575(CHEMBL3903475)
Affinity DataEC50:  38nMAssay Description:Agonist activity at human GPR142 expressed in CHO cells measured for 3 to 5 mins by Fluo-4AM dye-based FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/1/2018
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 142(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50201573(CHEMBL3908606)
Affinity DataEC50:  40nMAssay Description:Agonist activity at human GPR142 expressed in CHO cells measured after 30 to 60 mins by IP-One assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/1/2018
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 142(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50544803(CHEMBL4642312)
Affinity DataEC50:  41nMAssay Description:Agonist activity at human GPR142 receptor expressed in HEK293 cells assessed as accumulation of inositol phosphate incubated for 1 hr followed by IP1...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 142(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50440704(CHEMBL2430981)
Affinity DataEC50:  42nMAssay Description:Agonist activity at human GPR142 expressed in HEK293 cells assessed as inositol phosphate accumulation using [3H]-inositol after 1 hr by scintillatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 142(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM332762(US10196385, Example 1 | Cis-(chiral)-N-[(2-[5-(1,4...)
Affinity DataEC50:  43nMAssay Description:Agonist activity at human GPR142 receptor expressed in HEK293 cells assessed as accumulation of inositol phosphate incubated for 1 hr followed by IP1...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 142(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM332762(US10196385, Example 1 | Cis-(chiral)-N-[(2-[5-(1,4...)
Affinity DataEC50:  43.5nMAssay Description:HEK293 cells expressing human GPR142 are maintained in DMEM supplemented with 10% FBS and 800 μg/ml G418 (Geneticin) at 37° C. and 5% CO2. The c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2019
Entry Details
US Patent

TargetProbable G-protein coupled receptor 142(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50558167(CHEMBL4798957)
Affinity DataIC50: 45nMAssay Description:Agonist activity at human GPR142 expressed in CHO cells measured for 3 mins by Fluo-4M dye based FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 142(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50544806(CHEMBL4639333)
Affinity DataEC50:  46nMAssay Description:Agonist activity at human GPR142 receptor expressed in HEK293 cells assessed as accumulation of inositol phosphate incubated for 1 hr followed by IP1...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 142(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50558171(CHEMBL4790150)
Affinity DataIC50: 48nMAssay Description:Agonist activity at human GPR142 expressed in CHO cells measured for 3 mins by Fluo-4M dye based FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 142(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50440712(CHEMBL2430978)
Affinity DataEC50:  49nMAssay Description:Agonist activity at human GPR142 expressed in HEK293 cells assessed as inositol phosphate accumulation using [3H]-inositol after 1 hr by scintillatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 142(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50544796(CHEMBL4641543)
Affinity DataEC50:  51nMAssay Description:Agonist activity at human GPR142 receptor expressed in HEK293 cells assessed as accumulation of inositol phosphate incubated for 1 hr followed by IP1...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 142(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50390601(CHEMBL2069581)
Affinity DataEC50:  52nMAssay Description:Agonist activity at human GPR142 expressed in HEK293 cells assessed as inositol phosphate accumulation using [3H]-inositol after 1 hr by scintillatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 142(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50440693(CHEMBL2430983)
Affinity DataEC50:  52nMAssay Description:Agonist activity at human GPR142 expressed in HEK293 cells assessed as inositol phosphate accumulation using [3H]-inositol after 1 hr by scintillatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
Displayed 1 to 50 (of 231 total ) | Next | Last >>
Jump to: