Compile Data Set for Download or QSAR
Report error Found 37 for UniProtKB: Q95J97
TargetcAMP-dependent protein kinase(Rabbit)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 6760BDBM6760(CHEMBL281948 | methyl (15S,16R,18R)-16-hydroxy-15-...)
Affinity DataIC50: 0.0160nMAssay Description:Inhibition of cAMP dependent Protein kinase A of rabbit Skeletal Muscle.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetcAMP-dependent protein kinase(Rabbit)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 36603BDBM36603(4'',6''-Dideoxybalanol, 6)
Affinity DataKi:  3.40nM ΔG°:  -49.1kJ/mole IC50: 5.5nMpH: 7.5 T: 2°CAssay Description:Cyclic AMP-dependent protein kinase (PKA) enzyme inhibition assay using purified recombinant C subunit of PKA (catalytic (C) subunit (cPKA)) with hol...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2011
Entry Details Article
PubMed
TargetcAMP-dependent protein kinase(Rabbit)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 36604BDBM36604(5'-Deoxybalanol, 7)
Affinity DataKi:  3.5nM ΔG°:  -49.1kJ/mole IC50: 5.70nMpH: 7.5 T: 2°CAssay Description:Cyclic AMP-dependent protein kinase (PKA) enzyme inhibition assay using purified recombinant C subunit of PKA (catalytic (C) subunit (cPKA)) with hol...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2011
Entry Details Article
PubMed
TargetcAMP-dependent protein kinase(Rabbit)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 3207BDBM3207(CHEMBL193697 | 2-{[2,6-dihydroxy-4-({[(3R,4R)-3-[(...)
Affinity DataKi:  3.90nM ΔG°:  -48.8kJ/mole IC50: 6.30nMpH: 7.5 T: 2°CAssay Description:Cyclic AMP-dependent protein kinase (PKA) enzyme inhibition assay using purified recombinant C subunit of PKA (catalytic (C) subunit (cPKA)) with hol...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2011
Entry Details Article
PubMed
TargetcAMP-dependent protein kinase(Rabbit)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 3149BDBM3149(Acyclic Balanol Analog (-)-1 | 2-{[2,6-dihydroxy-4...)
Affinity DataKi:  4.70nM ΔG°:  -48.3kJ/molepH: 7.5 T: 2°CAssay Description:Cyclic AMP-dependent protein kinase (PKA) enzyme inhibition assay using purified recombinant C subunit of PKA (catalytic (C) subunit (cPKA)) with hol...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2011
Entry Details Article
PubMed
TargetcAMP-dependent protein kinase(Rabbit)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50058332BDBM50058332(methyl 10,23-di(ethylsulfanylmethyl)-16-hydroxy-15...)
Affinity DataIC50: 10nMAssay Description:Inhibition of cAMP dependent Protein kinase A of rabbit Skeletal Muscle.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetcAMP-dependent protein kinase(Rabbit)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 36602BDBM36602(14''-Decarboxybalanol hydrochloride, 5)
Affinity DataKi:  11nM ΔG°:  -46.2kJ/mole IC50: 18nMpH: 7.5 T: 2°CAssay Description:Cyclic AMP-dependent protein kinase (PKA) enzyme inhibition assay using purified recombinant C subunit of PKA (catalytic (C) subunit (cPKA)) with hol...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2011
Entry Details Article
PubMed
TargetcAMP-dependent protein kinase(Rabbit)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 2579BDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataKi:  35nMpH: 7.5Assay Description:Cyclic AMP-dependent protein kinase (PKA) enzyme inhibition assay using purified recombinant C subunit of PKA (catalytic (C) subunit (cPKA)) with hol...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2011
Entry Details Article
PubMed
TargetcAMP-dependent protein kinase(Rabbit)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 36606BDBM36606(H-89, 10)
Affinity DataKi:  48nMpH: 7.5Assay Description:Cyclic AMP-dependent protein kinase (PKA) enzyme inhibition assay using purified recombinant C subunit of PKA (catalytic (C) subunit (cPKA)) with hol...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2011
Entry Details Article
PubMed
TargetcAMP-dependent protein kinase(Rabbit)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 36605BDBM36605(KT5720, 9)
Affinity DataKi:  56nMpH: 7.5Assay Description:Cyclic AMP-dependent protein kinase (PKA) enzyme inhibition assay using purified recombinant C subunit of PKA (catalytic (C) subunit (cPKA)) with hol...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2011
Entry Details Article
PubMed
TargetcAMP-dependent protein kinase(Rabbit)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 15210BDBM15210(N-[2-(methylamino)ethyl]isoquinoline-5-sulfonamide...)
Affinity DataKi:  1.20E+3nMAssay Description:Inhibitory constant against cAPK (PKA)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetcAMP-dependent protein kinase(Rabbit)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50366348BDBM50366348(CHEMBL1233654)
Affinity DataKi:  3.00E+3nMAssay Description:Inhibitory constant against cAPK (PKA)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50169892BDBM50169892(3-{4-[4-(3-Chloro-phenylamino)-[1,3,5]triazin-2-yl...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Cyclin-dependent kinase 1-cyclin BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetcAMP-dependent protein kinase(Rabbit)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 36600BDBM36600(Benzophenone fragment, 2)
Affinity DataKi: >1.00E+4nM ΔG°: >-29.0kJ/molepH: 7.5 T: 2°CAssay Description:Cyclic AMP-dependent protein kinase (PKA) enzyme inhibition assay using purified recombinant C subunit of PKA (catalytic (C) subunit (cPKA)) with hol...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2011
Entry Details Article
PubMed
TargetcAMP-dependent protein kinase(Rabbit)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 36601BDBM36601(Hexahydroazepine, 3)
Affinity DataKi: >1.00E+4nMpH: 7.5Assay Description:Cyclic AMP-dependent protein kinase (PKA) enzyme inhibition assay using purified recombinant C subunit of PKA (catalytic (C) subunit (cPKA)) with hol...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2011
Entry Details Article
PubMed
TargetcAMP-dependent protein kinase(Rabbit)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 2672BDBM2672(6,7,12,13-Tetrahydro-5,7-dioxo-5H-indolo[2,3-a]pyr...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibitory activity was determined against protein kinase A (PKA) of rabbitMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetcAMP-dependent protein kinase(Rabbit)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 2583BDBM2583(bis-indolylmaleimide deriv. 8a | 3,4-bis(1H-indol-...)
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibitory activity was determined against protein kinase A (PKA) of rabbitMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetcAMP-dependent protein kinase(Rabbit)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50040914BDBM50040914(5-(4-Methoxy-phenylamino)-6-phenylamino-isoindole-...)
Affinity DataIC50: 5.00E+5nMAssay Description:Inhibitory activity was determined against protein kinase A (PKA) of rabbitMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetcAMP-dependent protein kinase(Rabbit)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50040925BDBM50040925(5,6-Bis-(4-methoxy-phenylamino)-isoindole-1,3-dion...)
Affinity DataIC50: 5.00E+5nMAssay Description:Inhibitory activity was determined against protein kinase A (PKA) of rabbitMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetcAMP-dependent protein kinase(Rabbit)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50040930BDBM50040930(5,6-Bis-(4-fluoro-phenylamino)-isoindole-1,3-dione...)
Affinity DataIC50: 5.00E+5nMAssay Description:Inhibitory activity was determined against protein kinase A (PKA) of rabbitMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetcAMP-dependent protein kinase(Rabbit)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50040926BDBM50040926(4,5-Bis-phenylamino-phthalic acid dimethyl ester |...)
Affinity DataIC50: 5.00E+5nMAssay Description:Inhibitory activity was determined against protein kinase A (PKA) of rabbitMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetcAMP-dependent protein kinase(Rabbit)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50040920BDBM50040920(5,6-Bis-p-tolylamino-isoindole-1,3-dione | CHEMBL7...)
Affinity DataIC50: 5.00E+5nMAssay Description:Inhibitory activity was determined against protein kinase A (PKA) of rabbitMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetcAMP-dependent protein kinase(Rabbit)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50040915BDBM50040915(5,6-Bis-(4-iodo-phenylamino)-isoindole-1,3-dione |...)
Affinity DataIC50: 5.00E+5nMAssay Description:Inhibitory activity was determined against protein kinase A (PKA) of rabbitMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetcAMP-dependent protein kinase(Rabbit)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50040921BDBM50040921(5,6-Bis-(4-diethylamino-phenylamino)-isoindole-1,3...)
Affinity DataIC50: 5.00E+5nMAssay Description:Inhibitory activity was determined against protein kinase A (PKA) of rabbitMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetcAMP-dependent protein kinase(Rabbit)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50040918BDBM50040918(5,6-Bis-(methyl-phenyl-amino)-isoindole-1,3-dione ...)
Affinity DataIC50: 5.00E+5nMAssay Description:Inhibitory activity was determined against protein kinase A (PKA) of rabbitMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetcAMP-dependent protein kinase(Rabbit)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50040913BDBM50040913(1,4-Diphenyl-1,2,3,4-tetrahydro-pyrrolo[3,4-g]quin...)
Affinity DataIC50: 5.00E+5nMAssay Description:Inhibitory activity was determined against protein kinase A (PKA) of rabbitMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetcAMP-dependent protein kinase(Rabbit)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50040917BDBM50040917(5-(Methyl-phenyl-amino)-6-phenylamino-isoindole-1,...)
Affinity DataIC50: 5.00E+5nMAssay Description:Inhibitory activity was determined against protein kinase A (PKA) of rabbitMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetcAMP-dependent protein kinase(Rabbit)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50040916BDBM50040916(5,6-Bis-(4-hydroxy-phenylamino)-isoindole-1,3-dion...)
Affinity DataIC50: 5.00E+5nMAssay Description:Inhibitory activity was determined against protein kinase A (PKA) of rabbitMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetcAMP-dependent protein kinase(Rabbit)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50040923BDBM50040923(N-Methyl-4,5-dianilinophthalimide | 2-Methyl-5,6-b...)
Affinity DataIC50: 5.00E+5nMAssay Description:Inhibitory activity was determined against protein kinase A (PKA) of rabbitMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetcAMP-dependent protein kinase(Rabbit)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50040927BDBM50040927(N-(1,3-Dioxo-6-phenylamino-2,3-dihydro-1H-isoindol...)
Affinity DataIC50: 5.00E+5nMAssay Description:Inhibitory activity was determined against protein kinase A (PKA) of rabbitMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetcAMP-dependent protein kinase(Rabbit)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50040922BDBM50040922(2-Phenyl-5,6-bis-phenylamino-isoindole-1,3-dione |...)
Affinity DataIC50: 5.00E+5nMAssay Description:Inhibitory activity was determined against protein kinase A (PKA) of rabbitMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetcAMP-dependent protein kinase(Rabbit)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50040912BDBM50040912(5,6-Bis-cyclohexylamino-isoindole-1,3-dione | CHEM...)
Affinity DataIC50: 5.00E+5nMAssay Description:Inhibitory activity was determined against protein kinase A (PKA) of rabbitMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetcAMP-dependent protein kinase(Rabbit)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50040931BDBM50040931(4,5-Bis-(4-fluoro-phenylamino)-phthalic acid dimet...)
Affinity DataIC50: 5.00E+5nMAssay Description:Inhibitory activity was determined against protein kinase A (PKA) of rabbitMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetcAMP-dependent protein kinase(Rabbit)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50040929BDBM50040929(5,6-bis(phenylamino)-1H-isoindole-1,3(2H)-dione | ...)
Affinity DataIC50: 5.00E+5nMAssay Description:Inhibitory activity was determined against protein kinase A (PKA) of rabbitMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetcAMP-dependent protein kinase(Rabbit)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50040924BDBM50040924(5,6-Bis-phenylsulfanyl-isoindole-1,3-dione | CHEMB...)
Affinity DataIC50: 5.00E+5nMAssay Description:Inhibitory activity was determined against protein kinase A (PKA) of rabbitMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetcAMP-dependent protein kinase(Rabbit)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50040919BDBM50040919(5,6-Bis-(biphenyl-4-ylamino)-isoindole-1,3-dione |...)
Affinity DataIC50: 5.00E+5nMAssay Description:Inhibitory activity was determined against protein kinase A (PKA) of rabbitMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetcAMP-dependent protein kinase(Rabbit)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50040928BDBM50040928(4-[6-(4-cyanoanilino)-1,3-dioxo-2,3-dihydro-1H-5-i...)
Affinity DataIC50: 5.00E+5nMAssay Description:Inhibitory activity was determined against protein kinase A (PKA) of rabbitMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed