Affinity DataIC50: 7.40nMAssay Description:Inhibition of YTHDC1 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
Affinity DataKd: 30nMAssay Description:Binding affinity to YTHDC1 (unknown origin) assessed as dissociation constantMore data for this Ligand-Target Pair
Affinity DataKd: 49nMAssay Description:Binding affinity to YTHDC1 (unknown origin) assessed as equilibrium dissociation constant by ITC analysisMore data for this Ligand-Target Pair
Affinity DataKd: 146nMAssay Description:Binding affinity to YTHDC1 (unknown origin) assessed as equilibrium dissociation constant by ITC analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 180nMAssay Description:Inhibition of GST-tagged YTHDC1 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
Affinity DataIC50: 350nMAssay Description:Inhibition of GST-tagged YTHDC1 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
Affinity DataIC50: 450nMAssay Description:Inhibition of GST-tagged YTHDC1 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
Affinity DataIC50: 460nMAssay Description:Inhibition of GST-tagged YTHDC1 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
Affinity DataIC50: 510nMAssay Description:Inhibition of GST-tagged YTHDC1 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
Affinity DataIC50: 590nMAssay Description:Inhibition of GST-tagged YTHDC1 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
Affinity DataIC50: 870nMAssay Description:Inhibition of GST-tagged YTHDC1 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
Affinity DataIC50: 960nMAssay Description:Inhibition of GST-tagged YTHDC1 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
Affinity DataIC50: 970nMAssay Description:Inhibition of GST-tagged YTHDC1 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of GST-tagged YTHDC1 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of GST-tagged YTHDC1 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of GST-tagged YTHDC1 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of GST-tagged YTHDC1 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of YTHDC1 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKd: 1.68E+3nMAssay Description:Binding affinity to YTHDC1 (unknown origin) assessed as dissociation constantMore data for this Ligand-Target Pair
Affinity DataKd: 1.70E+3nMAssay Description:Binding affinity to YTHDC1 (unknown origin) assessed as dissociation constantMore data for this Ligand-Target Pair
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of GST-tagged YTHDC1 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of GST-tagged YTHDC1 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of GST-tagged YTHDC1 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of GST-tagged YTHDC1 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of GST-tagged YTHDC1 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of YTHDC1 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of GST-tagged YTHDC1 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of GST-tagged YTHDC1 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of GST-tagged YTHDC1 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of GST-tagged YTHDC1 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of GST-tagged YTHDC1 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of GST-tagged YTHDC1 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of GST-tagged YTHDC1 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
Affinity DataIC50: 5.50E+3nMAssay Description:Inhibition of YTHDC1 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibition of GST-tagged YTHDC1 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
Affinity DataIC50: 8.00E+3nMAssay Description:Inhibition of GST-tagged YTHDC1 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
Affinity DataIC50: 9.00E+3nMAssay Description:Inhibition of GST-tagged YTHDC1 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
Affinity DataIC50: 9.00E+3nMAssay Description:Inhibition of GST-tagged YTHDC1 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.10E+4nMAssay Description:Inhibition of GST-tagged YTHDC1 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.10E+4nMAssay Description:Inhibition of GST-tagged YTHDC1 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.30E+4nMAssay Description:Inhibition of GST-tagged YTHDC1 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of GST-tagged YTHDC1 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
Affinity DataKd: 2.20E+4nMAssay Description:Binding affinity to YTHDC1 (unknown origin) assessed as dissociation constantMore data for this Ligand-Target Pair
Affinity DataIC50: 3.70E+4nMAssay Description:Inhibition of YTHDC1 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 3.90E+4nMAssay Description:Inhibition of YTHDC1 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 3.90E+4nMAssay Description:Binding affinity to GST-tagged YTHDC1 m6A-reader domain (unknown origin) using RRACH-containing methylated oligoRNA incubated for 3 hrs by HTRF assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3.90E+4nMAssay Description:Inhibition of YTHDC1 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 4.70E+4nMAssay Description:Inhibition of GST-tagged YTHDC1 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
Affinity DataKd: 5.80E+4nMAssay Description:Binding affinity to YTHDC1 (unknown origin) assessed as dissociation constantMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of GST-tagged YTHDC1 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair


3D Structure (crystal)







































