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Targets Binding with 23 Compounds
Target Name
Affinity Link(s)
Article(s)
UniProt
Files
4-hydroxy-3-methylbut-2-enyl diphosphate reductase
Ki:
5
IC50:
21
2
6
2D
3D
TSV
7-dehydrocholesterol reductase
Ki:
6
IC50:
25
Kd:
1
5
6
2D
3D
TSV
Alcohol dehydrogenase 1C
Ki:
23
1
7
2D
3D
TSV
Autoinducer 2-binding periplasmic protein LuxP
IC50:
15
EC50:
20
4
1
2D
3D
TSV
Beta-hexosaminidase subunit alpha/beta
Ki:
20
IC50:
3
3
6
2D
3D
TSV
Chitin synthase 3
IC50:
23
2
4
2D
3D
TSV
Cystathionine beta-lyase MetC
IC50:
23
1
3
2D
3D
TSV
Dehydrogenase/reductase SDR family member 9
IC50:
24
2
8
2D
3D
TSV
Dual specificity testis-specific protein kinase 2
IC50:
23
2
6
2D
3D
TSV
Ectonucleoside triphosphate diphosphohydrolase 3
Ki:
3
IC50:
21
6
6
2D
3D
TSV
Egl nine homolog 1/Prolyl hydroxylase EGLN2/Prolyl hydroxylase EGLN3/Transmembrane prolyl 4-hydroxylase
EC50:
46
1
18
2D
3D
TSV
Epidermal growth factor receptor [1-249,301-1210,T790M,L858R]
IC50:
23
1
18
2D
3D
TSV
Granzyme B
Ki:
23
3
4
2D
3D
TSV
Group IID secretory phospholipase A2
IC50:
38
3
9
2D
3D
TSV
GTPase KRas [1-169,G12D]
IC50:
24
1
7
2D
3D
TSV
Hypoxanthine phosphoribosyltransferase
Ki:
23
1
1
2D
3D
TSV
Interleukin-17F
IC50:
23
2
6
2D
3D
TSV
Metalloproteinase inhibitor 2
IC50:
23
1
1
2D
3D
TSV
Non-receptor tyrosine-protein kinase TYK2 [5-1181]
IC50:
31
4
6
2D
3D
TSV
NPC intracellular cholesterol transporter 1
EC50:
23
2
4
2D
3D
TSV
Phosphoenolpyruvate carboxykinase, cytosolic [GTP]
Ki:
7
IC50:
21
EC50:
9
3
7
2D
3D
TSV
Pleiotropic ABC efflux transporter of multiple drugs
IC50:
23
1
3
2D
3D
TSV
Protein farnesyltransferase alpha subunit/subunit beta
IC50:
23
1
2
2D
3D
TSV
Protein kinase C alpha/beta/gamma type
IC50:
23
2
7
2D
3D
TSV
RAF proto-oncogene serine/threonine-protein kinase [1-324]
IC50:
65
3
6
2D
3D
TSV
Receptor-type tyrosine-protein kinase FLT3 [N841I]
Kd:
23
2
7
2D
3D
TSV
Serine/threonine-protein kinase PknA
Ki:
23
1
5
2D
3D
TSV
Sodium/potassium-transporting ATPase subunit alpha-4/beta-1
IC50:
23
1
3
2D
3D
TSV
Solute carrier family 28 member 3
Ki:
23
IC50:
3
2
7
2D
3D
TSV
Solute carrier organic anion transporter family member 1A1
Ki:
24
5
1
2D
3D
TSV
Structural polyprotein
EC50:
31
1
4
2D
3D
TSV
Sulfotransferase 1E1
Ki:
8
IC50:
15
4
5
2D
3D
TSV
Trp operon repressor
Kd:
24
1
4
2D
3D
TSV
Tyrosine-protein kinase Lck [245-498]
IC50:
23
1
11
2D
3D
TSV
Ubiquitin carboxyl-terminal hydrolase isozyme L5
IC50:
23
4
9
2D
3D
TSV
VHL complex
Kd:
23
1
23
2D
3D
TSV
Zinc finger protein Helios
EC50:
25
1
10
2D
3D
TSV