PMID

Data

Article Title

Organization

An insight on synthetic and medicinal aspects of pyrazolo[1,5-a]pyrimidine scaffold.

University of Kwazulu-Natal

Azaflavones compared to flavones as ligands to the benzodiazepine binding site of brain GABA(A) receptors.

Lund University

Identification of anxiolytic/nonsedative agents among indol-3-ylglyoxylamides acting as functionally selective agonists at the gamma-aminobutyric acid-A (GABAA) alpha2 benzodiazepine receptor.

Universita Di Pisa

Synthesis of GABAA receptor agonists and evaluation of their alpha-subunit selectivity and orientation in the GABA binding site.

Johannes Gutenberg University

β-Carboline as a Privileged Scaffold for Multitarget Strategies in Alzheimer's Disease Therapy.

Univ. Grenoble Alpes

Synthesis and binding properties of MK-801 isothiocyanates; (+)-3-isothiocyanato-5-methyl-10,11-dihydro-5H-dibenzo[a,d]cyclohepten- 5,10-imine hydrochloride: a new, potent and selective electrophilic affinity ligand for the NMDA receptor-coupled phencyclidine binding site.

National Institute of Diabetes and Digestive and Kidney Diseases

Synthesis of alkyl-substituted arecoline derivatives as gamma-aminobutyric acid uptake inhibitors.

TBA

SL651498: an anxioselective compound with functional selectivity for alpha2- and alpha3-containing gamma-aminobutyric acid(A) (GABA(A)) receptors.

Sanofi Synthelabo

Characterization of the anxiolytic properties of a novel neuroactive steroid, Co 2-6749 (GMA-839; WAY-141839; 3alpha, 21-dihydroxy-3beta-trifluoromethyl-19-nor-5beta-pregnan-20-one), a selective modulator of gamma-aminobutyric acid(A) receptors.

Cocensys