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20 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
Structure-activity relationship studies on 1-(2-oxopropyl)indole-5-carboxylic acids acting as inhibitors of cytosolic phospholipase AEBI
University of M£Nster
Design, synthesis, and biological evaluation of 3-(1-Aryl-1H-indol-5-yl)propanoic acids as new indole-based cytosolic phospholipase A2a inhibitors.EBI
Asubio Pharma
Inhibition of group IVA cytosolic phospholipase A2 by thiazolyl ketones in vitro, ex vivo, and in vivo.EBI
University of Athens
1-(5-Carboxyindol-1-yl)propan-2-ones as inhibitors of human cytosolic phospholipase A2alpha: synthesis and properties of bioisosteric benzimidazole, benzotriazole and indazole analogues.EBI
University of M£Nster
1-(2-Carboxyindol-5-yloxy)propan-2-ones as inhibitors of human cytosolic phospholipase A2alpha: synthesis, biological activity, metabolic stability, and solubility.EBI
University of M£Nster
1-Indol-1-yl-propan-2-ones and related heterocyclic compounds as dual inhibitors of cytosolic phospholipase A(2)alpha and fatty acid amide hydrolase.EBI
University of M£Nster
Reactions of functionalized sulfonamides: application to lowering the lipophilicity of cytosolic phospholipase A2alpha inhibitors.EBI
Wyeth Research
 
Dicarboxylic acid inhibitors of phospholipase A2EBI
TBA
Inhibitory effect of synthetic C-C biflavones on various phospholipase A(2)s activity.EBI
Yeungnam University
1-(5-Carboxy- and 5-carbamoylindol-1-yl)propan-2-ones as inhibitors of human cytosolic phospholipase A2alpha: bioisosteric replacement of the carboxylic acid and carboxamide moiety.EBI
University of MüNster
Discovery of Ecopladib, an indole inhibitor of cytosolic phospholipase A2alpha.EBI
Wyeth Research
Design and synthesis of 1-indol-1-yl-propan-2-ones as inhibitors of human cytosolic phospholipase A2alpha.EBI
University of MüNster
1,2,4-Oxadiazolidin-3,5-diones and 1,3,5-triazin-2,4,6-triones as cytosolic phospholipase A2alpha inhibitors.EBI
Wyeth Research
Inhibition of cytosolic phospholipase A2alpha: hit to lead optimization.EBI
Wyeth Research
Structure-activity relationships of indole cytosolic phospholipase A(2)alpha inhibitors: substrate mimetics.EBI
Wyeth Research
Pyrrolidine inhibitors of human cytosolic phospholipase A(2).EBI
Shionogi
Substrate-Specific Inhibition Constants for Phospholipase AEBI
University of California
?-Lactones: A Novel Class of CaEBI
National and Kapodistrian University of Athens
Synthesis and characterization of 3-arylquinazolinone and 3-arylquinazolinethione derivatives as selective estrogen receptor beta modulators.BDB
Bristol-Myers Squibb
Discovery and evaluation of 3-(5-thien-3-ylpyridin-3-yl)-1H-indoles as a novel class of KDR kinase inhibitors.BDB
Merck Research Laboratories