26 articles for thisTarget
The following articles (labelled with PubMed ID or TBD) are for your review
Synthesis and structure-activity relationships of potent conformationally restricted retinoid X receptor ligands
Synthesis and receptor binding affinity of conformationally restricted retinoic acid analogues
Synthesis of highly potent RXR-specific retinoids: The use of a cyclopropyl group as a double bond isostere
Differential RXR & RAR activity of stilbene retinoid analogs bearing thiazole and imidazole carboxylic acids
Replacing alkyl sulfonamide with aromatic sulfonamide in sulfonamide-type RXR agonists favors switch towards antagonist activity.
Okayama University Graduate School Of Medicine
Aza-retinoids as novel retinoid X receptor-specific agonists.
Oxaprozin Analogues as Selective RXR Agonists with Superior Properties and Pharmacokinetics.
Design, synthesis and structure-activity relationship of novel RXR-selective modulators.
Design and synthesis of novel RXR-selective modulators with improved pharmacological profile.
Retinoic acid receptor ligands based on the 6-cyclopropyl-2,4-hexadienoic acid.
An improved synthesis of the C-linked glucuronide of N-(4-hydroxyphenyl)retinamide.
The Ohio State University
Enantioselective syntheses of potent retinoid X receptor ligands: differential biological activities of individual antipodes.
Tuning Nuclear Receptor Selectivity of Wy14,643 towards Selective Retinoid X Receptor Modulation.
Goethe University Frankfurt
Structure-activity relationship studies of novel heteroretinoids: induction of apoptosis in the HL-60 cell line by a novel isoxazole-containing heteroretinoid.
Stereoselective synthesis and receptor activity of conformationally defined retinoid X receptor selective ligands.
Synthesis of retinoid X receptor-specific ligands that are potent inducers of adipogenesis in 3T3-L1 cells.
Computer-Assisted Discovery and Structural Optimization of a Novel Retinoid X Receptor Agonist Chemotype.
Regulation of retinoidal actions by diazepinylbenzoic acids. Retinoid synergists which activate the RXR-RAR heterodimers.
University Of Tokyo
Synthesis and structure-activity relationships of retinoid X receptor selective diaryl sulfide analogs of retinoic acid.
A Novel Biphenyl-based Chemotype of Retinoid X Receptor Ligands Enables Subtype and Heterodimer Preferences.
Identification of the first retinoid X, receptor homodimer antagonist.
Discovery of novel retinoic acid receptor agonists having potent antiproliferative activity in cervical cancer cells.
Synthesis of high specific activity [3H]-9-cis-retinoic acid and its application for identifying retinoids with unusual binding properties.
Conformational effects on retinoid receptor selectivity. 2. Effects of retinoid bridging group on retinoid X receptor activity and selectivity.
Computer-Assisted Discovery of Retinoid X Receptor Modulating Natural Products and Isofunctional Mimetics.
Swiss Federal Institute Of Technology (Eth)
Natural-Products-Inspired Use of the gem-Dimethyl Group in Medicinal Chemistry.
St. John'S University