BDBM27658 1-(5-{[(2S)-2-aminopropanamido]methyl}thiophen-3-yl)-N-(pyridin-2-ylmethyl)-3-(trifluoromethyl)-1H-pyrazole-5-carboxamide::pyrazole scaffold, 7g
SMILES C[C@H](N)C(=O)NCc1cc(cs1)-n1nc(cc1C(=O)NCc1ccccn1)C(F)(F)F
InChI Key InChIKey=SEZBKGHSFWLPFK-NSHDSACASA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 27658
Affinity DataIC50: 3.35E+3nMpH: 9.0 T: 2°CAssay Description:Histone H3 is used as the substrate for CARM-1 enzyme, and the methylation is monitored using tritiated S-Adenosyl-Methionine (SAM) as a methyl donor...More data for this Ligand-Target Pair