BDBM402603 2-(1,4-diazepan-1-yl)-N- [3-(difluoromethyl)-1- methyl-1H-pyrazol-4- yl]pyrrolo[2,1- f][1,2,4]triazine-7- carboxamide trifluoroacetate::US10329295, Example 15
SMILES Cn1cc(NC(=O)c2ccc3cnc(nn23)N2CCCNCC2)c(n1)C(F)F
InChI Key InChIKey=JEJYMFZUCMPIHO-UHFFFAOYSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 402603
Affinity DataIC50: 6nMAssay Description:The kinase activity of IRAK4 is determined by its ability to catalyze the phosphorylation of a fluorescent polypeptide substrate. The extent of phosp...More data for this Ligand-Target Pair