BDBM50142759 (R)-N-(4-(1-(3-(4-tert-butylbenzyl)thioureido)ethyl)phenyl)methanesulfonamide::CHEMBL412885::N-(4-tert-butylbenzyl)-N'-{(1R)-1-[4-(methylsulfonylamino)phenyl]ethyl}thiourea::N-(4-{(R)-1-[3-(4-tert-Butyl-benzyl)-thioureido]-ethyl}-phenyl)-methanesulfonamide
SMILES C[C@@H](NC(=S)NCc1ccc(cc1)C(C)(C)C)c1ccc(NS(C)(=O)=O)cc1
InChI Key InChIKey=MRGDOZGZFFCDRJ-OAHLLOKOSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 4 hits for monomerid = 50142759
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Sookmyung Women'S University
Curated by ChEMBL
Sookmyung Women'S University
Curated by ChEMBL
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at TRPV1 in Sprague-Dawley rat DRG neuron assessed as intracellular 45Ca2+ influx by scintillation countingMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Sookmyung Women'S University
Curated by ChEMBL
Sookmyung Women'S University
Curated by ChEMBL
Affinity DataIC50: 50nMAssay Description:Antagonist activity at TRPV1 in neonatal rat DRG neurons assessed as inhibition of capsaicin-induced intracellular calcium after 10 mins in presence ...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Sookmyung Women'S University
Curated by ChEMBL
Sookmyung Women'S University
Curated by ChEMBL
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at TRPV1 in neonatal rat DRG neurons assessed as increase in calcium influx after 10 mins in presence of 45Ca2+ by Beckman CP scinti...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Sookmyung Women'S University
Curated by ChEMBL
Sookmyung Women'S University
Curated by ChEMBL
Affinity DataIC50: 50nMAssay Description:Antagonist activity at TRPV1 in Sprague-Dawley rat DRG neuron assessed as reduction of capsaicin-stimulated intracellular 45Ca2+ influx by scintillat...More data for this Ligand-Target Pair