BDBM379363 5-((4-(cyclopropylamino)-5-(trifluoromethyl)pyrimidin-2-yl)amino)indolin-2-one::US10266549, Example 240::US10774092, Example 240
SMILES FC(F)(F)c1cnc(Nc2ccc3NC(=O)Cc3c2)nc1NC1CC1
InChI Key InChIKey=LSEXUJNSJCGXHK-UHFFFAOYSA-N
Data 2 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 379363
Affinity DataIC50: <200nMAssay Description:ULK1 inhibition assay is a screening assay to identify compounds that inhibit kinase activity of ULK1 using the ULKtide peptide. In some embodiments,...More data for this Ligand-Target Pair