BDBM50583753 CHEMBL5088511

SMILES Cc1nc2ccc(nc2n1CCOc1ccccc1)-c1cc(N)nc(N)c1

InChI Key InChIKey=XQMMPFLQOCIGRW-UHFFFAOYSA-N

Data  4 IC50

PDB links: 1 PDB ID matches this monomer.

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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50583753   

TargetDual specificity tyrosine-phosphorylation-regulated kinase 2(Homo sapiens (Human))
Servier Research Institute Of Medicinal Chemistry

Curated by ChEMBL
LigandPNGBDBM50583753(CHEMBL5088511)
Affinity DataIC50:  9nMAssay Description:Inhibition of DYRK2 (unknown origin) using Ulight-MBP as substrate and ATP as co-substrate incubated for 40 mins and measured after 1 hr by TR-FRET a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed