BDBM317009 Propane-1-sulfonic acid {2,4- difluoro-3-[4-(oxetan-3- ylamino)-7H-pyrrolo[2,3- d]pyrimidine-5-carbonyl]- phenyl}-amide::US9617267, Compound P-1060

SMILES CCCS(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncnc(NC4COC4)c23)c1F

InChI Key InChIKey=GGPYYUMXGVJJGG-UHFFFAOYSA-N

Data  9 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Similarity at least:  must be >=0.5
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 317009   

TargetEpidermal growth factor receptor [T790M,L858R](Homo sapiens (Human))
Plexxikon

US Patent
LigandPNGBDBM317009(Propane-1-sulfonic acid {2,4- difluoro-3-[4-(oxeta...)
Affinity DataIC50: <100nMAssay Description:Assays for biochemical and cell based activity are known in the art, for example, as described in PCT publication WO 2007/002433, the disclosure of w...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent