BDBM50158830 CHEMBL3785583

SMILES CC(C)c1c([nH]c2c(cnn2c1=O)C#N)-c1cnn(c1)C(C)(C)C

InChI Key InChIKey=KRXWJZIHQRIGSJ-UHFFFAOYSA-N

Data  13 IC50  2 EC50

PDB links: 1 PDB ID matches this monomer.

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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50158830   

TargetLysine-specific demethylase 5C(Homo sapiens (Human))TBA
LigandPNGBDBM50158830(CHEMBL3785583)
Affinity DataIC50:  66nMAssay Description:Inhibition of KDM5C (unknown origin ) by HTMS assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetLysine-specific demethylase 5C(Homo sapiens (Human))TBA
LigandPNGBDBM50158830(CHEMBL3785583)
Affinity DataIC50:  66nMAssay Description:Inhibition of KDM5C (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific demethylase 5C(Homo sapiens (Human))TBA
LigandPNGBDBM50158830(CHEMBL3785583)
Affinity DataIC50:  66nMAssay Description:Inhibition of KDM5C (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed