BDBM50572221 CHEMBL4862974
SMILES OC(=O)c1cc(c2cc(ccc2n1)N1CCC2(CC(=C2)c2c(onc2-c2c(Cl)cncc2Cl)C2CC2)CC1)C(F)(F)F
InChI Key InChIKey=WPGAVSDZYIRUGE-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 50572221
Affinity DataIC50: >4.00E+4nMAssay Description:Antagonist activity at human RORalpha (272 to 557 residues) co-expressed with Gal4-luciferase reporter in human Jurkat cells incubated for 18 hrs by ...More data for this Ligand-Target Pair
Affinity DataEC50: >4.00E+4nMAssay Description:Agonist activity at human RORalpha (272 to 557 residues) co-expressed with Gal4-luciferase reporter in human Jurkat cells incubated for 18 hrs by Ste...More data for this Ligand-Target Pair