BDBM264256 6-(2,6-Dichlorophenyl)-2-((4-(1-methylpiperidin-4-yl)phenyl)amino)pyrido[4,3-d]pyrimidin-5(6H)-one, HCl::US9714244, 10

SMILES CN1CCC(CC1)c1ccc(Nc2ncc3c(ccn(-c4c(Cl)cccc4Cl)c3=O)n2)cc1

InChI Key InChIKey=DFSAQPXRPWPPCR-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 264256   

TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Almac Discovery

US Patent
LigandPNGBDBM264256(6-(2,6-Dichlorophenyl)-2-((4-(1-methylpiperidin-4-...)
Affinity DataIC50:  105nMAssay Description:Compounds were tested for inhibition of the human ether a go-go related gene (hERG) K+ channel using IonWorks patch clamp electrophysiology at Essen ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent