BDBM50184778 CHEMBL3823711::US10294227, Code 540
SMILES COc1cc(ccc1NC(=O)NC(C)(C)C)-c1nn(CCN2CCC(CC2)N(C)C)c2ncnc(N)c12
InChI Key InChIKey=KZRDVFBPXXGSPD-UHFFFAOYSA-N
Data 17 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 50184778
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University Court of The University of Edinburgh
US Patent
University Court of The University of Edinburgh
US Patent
Affinity DataIC50: 550nMAssay Description:Compound IC50 values were determined from 10-point, 1:3 dilution curves starting at either 100 μM or 10 μM with 10 μM ATP, by Reaction...More data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University Court of The University of Edinburgh
US Patent
University Court of The University of Edinburgh
US Patent
Affinity DataIC50: 194nMAssay Description:Inhibition of C-terminal His-tagged full length human SRC expressed in insect cells preincubated for 20 mins using poly[Glu,Tyr]4:1 as substrate meas...More data for this Ligand-Target Pair