BDBM432225 N-[1-(4-Cyanophenyl)-1H-pyrazol-3-yl]-N-(1-methylpiperidin-4-yl)thiophene-2-::US10577360, Example 89
SMILES CN1CCC(CC1)N(C(=O)c1cccs1)c1ccn(n1)-c1ccc(cc1)C#N
InChI Key InChIKey=HORLRCMRIBAKMX-UHFFFAOYSA-N
Data 2 KI
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 432225
TargetVoltage-dependent calcium channel subunit alpha-2/delta-1(Homo sapiens (Human))
Esteve Pharmaceuticals
US Patent
Esteve Pharmaceuticals
US Patent
Affinity DataKi: 2.75E+3nMAssay Description:Human α2δ-1 enriched membranes (2.5 μg) were incubated with 15 nM of radiolabeled [3H]-Gabapentin in assay buffer containing Hepes-KOH...More data for this Ligand-Target Pair