BDBM289616 2-(((2S,6R)-2,6-Dimethylmorpholino)methyl)-4-(4-methoxybenzyl)pyrazolo[1,5-c]thieno[3,2-e]pyrimidin-5(4H)-one::US10092575, Example 104::US10376514, Example 184
SMILES COc1ccc(Cn2c3sc(CN4C[C@H](C)O[C@H](C)C4)cc3c3ccnn3c2=O)cc1
InChI Key InChIKey=UHDDFCNUWMNGAD-IYBDPMFKSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 289616
TargetDual specificity calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1B(Human)
Dart Neuroscience (Cayman)
US Patent
Dart Neuroscience (Cayman)
US Patent
Affinity DataEC50: 550nMT: 25°CAssay Description:The IMAP TR-FRET PDE assay was optimized for concentration of enzyme, Calmodulin, cAMP or cGMP substrate, DMSO tolerance, and incubation time. Into e...More data for this Ligand-Target Pair
TargetDual specificity calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1B(Human)
Dart Neuroscience (Cayman)
US Patent
Dart Neuroscience (Cayman)
US Patent
Affinity DataEC50: <100nMT: 25°CAssay Description:The IMAP TR-FRET PDE assay was optimized for concentration of enzyme, Calmodulin, cAMP or cGMP substrate, DMSO tolerance, and incubation time. Into e...More data for this Ligand-Target Pair