BDBM250488 US9464044, 121
SMILES NC(=O)C12CC3CC(C1)[C@H](NC(=O)c1cccc(NS(=O)(=O)c4ccc(F)cc4F)c1)C(C3)C2
InChI Key InChIKey=JPOAXBHNIKMLBX-CJEYPXOASA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 250488
Affinity DataIC50: 7.80nMpH: 6.0 T: 25°CAssay Description:The inhibiting activity of 11β-HSD1 derived from microsomal fractions was measured using the HTRF assay (62CO2PEB, Cisbio). Different concentrat...More data for this Ligand-Target Pair