BDBM50257037 CHEMBL103772::[3H]NGD-941

SMILES C(N1CCN(CC1)c1ncccn1)c1c[nH]c(n1)-c1ccccc1

InChI Key InChIKey=OTVQCHUIPJYASM-UHFFFAOYSA-N

Data  3 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 5 hits for monomerid = 50257037   

TargetD(4) dopamine receptor(Human)
University of North Carolina at Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50257037([3H]NGD-941 | CHEMBL103772)
Affinity DataKi:  4.30nMAssay Description:Displacement of 3H-N-Methylspiperone from DRD4 in human HEK293T cells membrane assessed as inhibition constant incubated for 2 hrs by radioligand com...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetD(2) dopamine receptor(Human)
University of North Carolina at Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50257037([3H]NGD-941 | CHEMBL103772)
Affinity DataKi:  36nMAssay Description:Displacement of 3H-N-Methylspiperone from DRD2 in human HEK293T cells membrane assessed as inhibition constant incubated for 2 hrs by radioligand com...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50257037([3H]NGD-941 | CHEMBL103772)
Affinity DataKi:  180nMAssay Description:Inhibition of serotonin 5-HT1A receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2019
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50257037([3H]NGD-941 | CHEMBL103772)
Affinity DataKi:  750nMAssay Description:Inhibition of serotonin 5-HT3 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2019
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
University of North Carolina at Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50257037([3H]NGD-941 | CHEMBL103772)
Affinity DataKi:  2.23E+3nMAssay Description:Inhibition of human dopamine D2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2019
Entry Details Article
PubMed