BDBM614811 A7-1-2::US20230271937, Example A7-1-2::US20230271937, Example A7-49

SMILES NC(=O)CN1CC[C@@H](CNc2ncnc(N(Cc3ccc(cc3)C(F)(F)F)C3CC3)c2F)[C@@H](O)C1

InChI Key InChIKey=ZJABFXPOYIJVMY-UHFFFAOYSA-N

Data  2 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 614811   

TargetPeroxisome proliferator-activated receptor gamma(Human)
Nuevolution

US Patent
LigandPNGBDBM614811(US20230271937, Example A7-1-2 | US20230271937, Exa...)
Affinity DataEC50:  1.5nMAssay Description:The HEK293 cell line is co-transfected transiently with two plasmids, one with the RORγ ligand-binding domain fused to galactose-responsive tran...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2023
Entry Details
US Patent

TargetPeroxisome proliferator-activated receptor gamma(Human)
Nuevolution

US Patent
LigandPNGBDBM614811(US20230271937, Example A7-1-2 | US20230271937, Exa...)
Affinity DataEC50:  168nMAssay Description:The HEK293 cell line is co-transfected transiently with two plasmids, one with the RORγ ligand-binding domain fused to galactose-responsive tran...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2023
Entry Details
US Patent