BDBM130924 US8829190, 102

SMILES COc1ccc(C(=O)Cc2c(Cl)cncc2Cl)n2ncnc12

InChI Key InChIKey=HOOKGSVYZWYNRS-UHFFFAOYSA-N

Data  2 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 130924   

TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Human)
TBA

Curated by ChEMBL

LigandBDBM130924(US8829190, 102)Copy SMILESCopy InChI

Affinity DataIC50: 100nMAssay Description:Inhibition of PDE4 (unknown origin)More data for this Ligand-Target Pair

Target InfoPDB
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sidSimilars

In Depth
Date in BDB:
3/22/2022
Entry Details Article
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TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A(Human)
Leo Pharma

US Patent

LigandBDBM130924(US8829190, 102)Copy SMILESCopy InChI

Affinity DataIC50: 134nMAssay Description:Human recombinant PDE4 (Gene bank accession no NM006203) was incubated for 1 hour with the test compound at concentrations up to 10 μM, with cAM...More data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sidSimilars

In Depth
Date in BDB:
2/16/2015
Entry Details
Copy BDB DOIUS Patent

Copy reaction URL