BDBM130939 US8829190, 117

SMILES COc1ccc(C(=O)Cc2c(Cl)cncc2Cl)n2nc(nc12)C1(CC1)C(=O)NC(C)C

InChI Key InChIKey=BSWGHDDDYLHRNH-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 130939   

TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A(Human)
Leo Pharma

US Patent
LigandPNGBDBM130939(US8829190, 117)
Affinity DataIC50: 0.200nMAssay Description:Human recombinant PDE4 (Gene bank accession no NM006203) was incubated for 1 hour with the test compound at concentrations up to 10 μM, with cAM...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/16/2015
Entry Details
US Patent