BDBM13236 5-N-(2-chloro-6-methylphenyl)-4-methyl-2-N-(thiophene-2-)-1,3-thiazole-2,5-diamido::BMS-354825 2-Amino-4-methyl-thiazole Analog 7j::N-(2-chloro-6-methylphenyl)-4-methyl-2-[(thien-2-ylcarbonyl)amino]-1,3-thiazole-5-carboxamide

SMILES Cc1nc(NC(=O)c2cccs2)sc1C(=O)Nc1c(C)cccc1Cl

InChI Key InChIKey=FKGOQKFINQMHDF-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 13236   

TargetTyrosine-protein kinase Lck(Human)
Bristol-Myers Squibb

LigandPNGBDBM13236(N-(2-chloro-6-methylphenyl)-4-methyl-2-[(thien-2-y...)
Affinity DataIC50: 130nMAssay Description:IC50 is the inhibitor concentration, which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-33P] lab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2007
Entry Details Article
PubMed