BDBM173111 US9096589, 1-(4-Chloro-phenyl)-2-{2-[2-(5,7-dimethyl-imidazo[1,2-a]pyrimidin-2-yl)-ethyl]-4-thiazol-5-yl-imidazol-1-yl}-ethanol

SMILES Cc1cc(C)n2cc(CCc3nc(cn3CC(O)c3ccc(Cl)cc3)-c3cncs3)nc2n1

InChI Key InChIKey=VBIPSTGQANQRON-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Similarity at least:  must be >=0.5
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 173111   

LigandPNGBDBM173111(US9096589, 1-(4-Chloro-phenyl)-2-{2-[2-(5,7-dimeth...)
Affinity DataIC50: 5.70nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2016
Entry Details
US Patent