BDBM177936 US9120797, 34
SMILES CN(C)C1(CCC2(CC1)NCCc1c2[nH]c2ccc(F)cc12)c1ccccc1
InChI Key InChIKey=JBRPRZXCKRICQC-UHFFFAOYSA-N
Data 2 KI
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 177936
Affinity DataKi: 0.700nM ΔG°: -12.5kcal/moleT: 25°CAssay Description:The receptor affinity for the human mu-opiate receptor was determined in a homogeneous batch in microtitre plates. For this, dilution series of the p...More data for this Ligand-Target Pair
Affinity DataKi: 1.40nM ΔG°: -12.1kcal/molepH: 7.4 T: 25°CAssay Description:The cyclohexane derivatives of the general formula I were investigated in a receptor binding assay with 3H-nociceptin/orphanin FQ with membranes from...More data for this Ligand-Target Pair