BDBM184357 US9150578, I-005

SMILES CN(C)C(=O)Cn1cc(Nc2ncc3CCc4nn(C)c(c4-c3n2)-c2ccc(cc2)-c2cnn(C)c2)cn1

InChI Key InChIKey=URABRDOUNMLPLA-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Similarity at least:  must be >=0.5
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 184357   

TargetInsulin receptor [964-1370](Human)
Boehringer Ingelheim International

US Patent
LigandPNGBDBM184357(US9150578, I-005)
Affinity DataIC50:  0.100nMpH: 7.4Assay Description:The kinase activity is measured by DELFIA.RTM. assay (dissociation-enhanced lanthanide fluorescence immunoassay, Perkin Elmer). The cytoplasmic kinas...More data for this Ligand-Target Pair
In DepthDetails US Patent