BDBM184387 US9150578, I-035

SMILES Cn1cc(cn1)-c1cccc(Cc2c-3c(CCc4cnc(Nc5ccn(CCCN6CCCC6)n5)nc-34)nn2C)c1

InChI Key InChIKey=WFXSEBKHQBTMMS-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 184387   

TargetInsulin receptor [964-1370](Human)
Boehringer Ingelheim International

US Patent
LigandPNGBDBM184387(US9150578, I-035)
Affinity DataIC50:  0.0800nMpH: 7.4Assay Description:The kinase activity is measured by DELFIA.RTM. assay (dissociation-enhanced lanthanide fluorescence immunoassay, Perkin Elmer). The cytoplasmic kinas...More data for this Ligand-Target Pair
In DepthDetails US Patent