BDBM184425 US9150578, I-059

SMILES COCCn1cc(cn1)-c1ccc(cc1)-c1c-2c(CCc3cnc(Nc4ccn(CCN(C)C)n4)nc-23)nn1C

InChI Key InChIKey=OWPFZNYKPFPFIT-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Similarity at least:  must be >=0.5
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 184425   

TargetInsulin receptor [964-1370](Human)
Boehringer Ingelheim International

US Patent
LigandPNGBDBM184425(US9150578, I-059)
Affinity DataIC50:  0.130nMpH: 7.4Assay Description:The kinase activity is measured by DELFIA.RTM. assay (dissociation-enhanced lanthanide fluorescence immunoassay, Perkin Elmer). The cytoplasmic kinas...More data for this Ligand-Target Pair
In DepthDetails US Patent