BDBM184486 US9150578, I-119

SMILES CCn1ccc(Nc2ncc3CCc4nn(C)c(c4-c3n2)-c2ccc(cc2)-c2cnn(CCN3CCC(CC3)N(C)C)c2)n1

InChI Key InChIKey=MRNCAMTZMKCLDO-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 184486   

TargetInsulin receptor [964-1370](Human)
Boehringer Ingelheim International

US Patent
LigandPNGBDBM184486(US9150578, I-119)
Affinity DataIC50:  0.0900nMpH: 7.4Assay Description:The kinase activity is measured by DELFIA.RTM. assay (dissociation-enhanced lanthanide fluorescence immunoassay, Perkin Elmer). The cytoplasmic kinas...More data for this Ligand-Target Pair
In DepthDetails US Patent