BDBM195767 US9670212, 143 N-{[2-(4-acetylpiperazin-1-yl)-8-methylquinolin-3-yl]methyl}-9H-purin-6-amine

SMILES CC(=O)N1CCN(CC1)c1nc2c(C)cccc2cc1CNc1ncnc2[nH]cnc12

InChI Key InChIKey=PYXANJKLSKNGGP-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 195767   

TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Human)
Exelixis

US Patent

LigandBDBM195767(US9670212, 143 N-{[2-(4-acetylpiperazin-1-yl)-8-me...)Copy SMILESCopy InChI

Affinity DataIC50: 50nMAssay Description:Kinase activity is measured as the percent of ATP consumed following the kinase reaction using luciferase-luciferin-coupled chemiluminescence. Reacti...More data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoKEGGPC cidPC sidSimilars

In Depth
Date in BDB:
7/7/2018
Entry Details
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