BDBM196846 US9212187, 330

SMILES CCN1c2ccc(CN(CCc3cccnc3)C(=O)Cc3cn(C)c4ccccc34)cc2N(C)C(=O)C(C)(C)C1=O

InChI Key InChIKey=PTHTUNQWYIDNJP-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Similarity at least:  must be >=0.5
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 196846   

TargetPotassium voltage-gated channel subfamily A member 5(Human)
Otsuka Pharmaceutical

US Patent
LigandPNGBDBM196846(US9212187, 330)
Affinity DataIC50: 860nMAssay Description:CHO-K1 cell lines stably expressing human Kv1.5 channels were prepared in the following manner.Full-length human Kv1.5 cDNA was cloned from a human h...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2016
Entry Details
US Patent