BDBM203317 US9242981, 46
SMILES CN1C[C@@H](NC(=O)N2CCc3[nH]nc(c3C2)-c2ccncc2)[C@@H](C1)c1ccccc1C
InChI Key
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 203317
Affinity DataIC50: 0.890nMAssay Description:Activated ERK2 activity was also determined in the IMAP assay format using the procedure outlined above. 1 μl of 25× compound was added to 14 ...More data for this Ligand-Target Pair
Affinity DataKd: 0.700nMT: 2°CAssay Description:The SAR (Structure Activity Relationship) for ERK ligands covered by
this invention was interrogated using the TdF (Temperature Dependence
Fluoresc...More data for this Ligand-Target Pair