BDBM204831 US9242977, 34

SMILES CCNc1ncc(s1)-c1ccc(Oc2ccc(NC(=O)Nc3cc(cnc3-c3ccc(C)c(C)c3)C(F)(F)F)cn2)cc1

InChI Key InChIKey=KPFPNNCNIXMYCQ-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 204831   

LigandPNGBDBM204831(US9242977, 34)
Affinity DataIC50:  6nMAssay Description:TrkA kinase-inhibiting activity in cell systems was measured using CHO-K1 cells expressing human TrkA and NFAT-bla (CellSenser TrkA-NFAT-bla CHO-K1 c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent

LigandPNGBDBM204831(US9242977, 34)
Affinity DataIC50:  180nMpH: 7.5Assay Description:TrkA-inhibiting activity was measured according to the following method using LanthaScreen kinase assay reagents (Invitrogen; Fluorescein-Poly GT, La...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent