BDBM23822 (2R)-2-amino-3-{[(4-methylphenyl)diphenylmethyl]sulfanyl}propanoic acid::S-Trityl-L-Cysteine (STLC) Analogue, 51
SMILES Cc1ccc(cc1)C(SC[C@H](N)C(O)=O)(c1ccccc1)c1ccccc1
InChI Key InChIKey=ZPXQDWLBSHVOEI-NRFANRHFSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 3 hits for monomerid = 23822
Affinity DataKi: 13.6nMAssay Description:Inhibition of N-terminal hexa-histidine tagged human cloned Eg5 (1 to 368 amino acids) expressed in Escherichia coli BL21 (DE3) assessed as reduction...More data for this Ligand-Target Pair
Affinity DataKi: 100nM ΔG°: -9.54kcal/moleT: 25°CAssay Description:The microtubule-activated ATPase rates were measured using the pyruvate kinase/lactate dehydrogenase-linked assay. To optimize the signal for basal E...More data for this Ligand-Target Pair
Affinity DataIC50: 61.7nMAssay Description:Inhibition of C-terminal His6-tagged human Eg5 microtubule-stimulated ATPase activityMore data for this Ligand-Target Pair