BDBM241610 US9409915, 79::US9718820, Compound 80
SMILES COc1c(nn(C)c1-c1nc2cc(nc(OC)c2[nH]1)-c1ccccc1C(F)(F)F)C(C)(C)C
InChI Key InChIKey=HSKWXHNAPILKQD-UHFFFAOYSA-N
Data 3 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 3 hits for monomerid = 241610
Affinity DataIC50: 20nMT: 37°CAssay Description:HEK293 cells stably expressing canine TRPM8 were routinely grown as monolayers in Dulbecco's minimum essential medium supplemented with 10% FBS, 2 mM...More data for this Ligand-Target Pair
Affinity DataIC50: 42nMT: 25°CAssay Description:HEK293 cells stably expressing canine TRPM8 were routinely grown as monolayers in Dulbecco's minimum essential medium supplemented with 10% FBS, ...More data for this Ligand-Target Pair
Affinity DataIC50: 20nMT: 25°CAssay Description:HEK293 cells stably expressing canine TRPM8 were routinely grown as monolayers in Dulbecco's minimum essential medium supplemented with 10% FBS, ...More data for this Ligand-Target Pair