BDBM242891 US9427442, 19

SMILES C[C@@H](C[C@@H]([C@@H](CCC(F)(F)F)C(=O)N[C@H]1N=C(c2ccccc2)c2cccc(F)c2NC1=O)C(N)=O)C(F)(F)F

InChI Key InChIKey=PNAKCIOOKPJNCG-HMVOWMFESA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 242891   

LigandPNGBDBM242891(US9427442, 19)
Affinity DataIC50:  2.40nMAssay Description:The Notch-CBF1 (C-promoter binding factor I) cell based transactivation assay is based on the ability of the released Notch intracellular domain frag...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent


LigandPNGBDBM242891(US9427442, 19)
Affinity DataIC50:  2.90nMAssay Description:The Notch-CBF1 (C-promoter binding factor I) cell based transactivation assay is based on the ability of the released Notch intracellular domain frag...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent