BDBM247410 US9453017, 2

SMILES C[C@@H](CN1CCC(n2c(=O)[nH]c3cc(Br)ccc32)CC1)NC(=O)[C@@H]1C[C@@H]1c1ccccc1

InChI Key InChIKey=JSVNNLRZCJAYTQ-UHFFFAOYSA-N

Data  4 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 247410   

TargetPhospholipase D1(Human)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 247410BDBM247410(US9453017, 2)
Affinity DataIC50: 15nMAssay Description:In vitro PLD activity is measured with an exogenous substrate assay as previously described (Brown, H. A. et al. (1993) Cell 75:1137-1144). Briefly, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
US Patent

TargetPhospholipase D2(Human)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 247410BDBM247410(US9453017, 2)
Affinity DataIC50: 1.10E+3nMAssay Description:In vitro PLD activity is measured with an exogenous substrate assay as previously described (Brown, H. A. et al. (1993) Cell 75:1137-1144). Briefly, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
US Patent