BDBM261733 1-fluoro-N-[(3S,4R)- 3-hydroxytetra- hydropyran-4-yl]-4- [[6-(1-methylpyrazol- 4-yl)-3-pyridyl]methyl]- naphthalene-2- carboxamide::US9708302, 19

SMILES Cn1cc(cn1)-c1ccc(Cc2cc(C(=O)N[C@@H]3CCOC[C@H]3O)c(F)c3ccccc23)cn1

InChI Key InChIKey=PQZBCCGOIMNBLV-DNQXCXABSA-N

Data  2 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 261733   

TargetMuscarinic acetylcholine receptor M1(RAT)
Hoffmann-La Roche

US Patent
LigandPNGBDBM261733(1-fluoro-N-[(3S,4R)- 3-hydroxytetra- hydropyran-4-...)
Affinity DataEC50:  97nMAssay Description:The assay is designed to select compounds that possess modulator activity at the acetylcholine muscarinic receptor expressed in CHO cells by measurin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM261733(1-fluoro-N-[(3S,4R)- 3-hydroxytetra- hydropyran-4-...)
Affinity DataEC50:  65nMAssay Description:The assay is designed to select compounds that possess modulator activity at the acetylcholine muscarinic receptor expressed in CHO cells by measurin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent