BDBM270586 (S)-N6- (benzo[d]thiazol-7- yl(1-(1- (trifluoromethyl) cyclopropyl)-1H-1,2,3- triazol-4-yl)methyl)- 8-bromo-N4- neopentylquinazoline- 4,6-diamine::US10059695, I-18::US10577352, Compound I-18
SMILES CC(C)(C)CNc1ncnc2c(Br)cc(N[C@H](c3cn(nn3)C3(CC3)C(F)(F)F)c3cccc4ncsc34)cc12
InChI Key InChIKey=LWKBAGGIOZPLOK-QFIPXVFZSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 4 hits for monomerid = 270586
Affinity DataIC50: 8nMpH: 7.0 T: 25°CAssay Description:EGFR activity was measured using KinEASE (Cisbio), a time-resolved fluorescence resonance energy transfer (TR-FRET) immunoassay. In this assay, EGFR-...More data for this Ligand-Target Pair
Affinity DataEC50: 195nMAssay Description:EGFR activity was measured using KinEASE (Cisbio), a time-resolved fluorescence resonance energy transfer (TR-FRET) immunoassay. In this assay, EGFR-...More data for this Ligand-Target Pair
Affinity DataIC50: 8nMAssay Description:EGFR activity was measured using KinEASE (Cisbio), a time-resolved fluorescence resonance energy transfer (TR-FRET) immunoassay. In this assay, EGFR-...More data for this Ligand-Target Pair
Affinity DataEC50: 195nMpH: 7.0 T: 25°CAssay Description:EGFR activity was measured using KinEASE (Cisbio), a time-resolved fluorescence resonance energy transfer (TR-FRET) immunoassay. In this assay, EGFR-...More data for this Ligand-Target Pair